Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50009832
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532608(CHEMBL4525688)
Affinity DataIC50: 1nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as blocking of inward/outward currents after 20 to 48 hrs in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532608(CHEMBL4525688)
Affinity DataIC50: 1nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as blocking of inward/outward currents after 20 to 48 hrs in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532612(CHEMBL4459054)
Affinity DataIC50: 1nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as reduction of rise in intracellular Ca2+ concentration after 60 to 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532612(CHEMBL4459054)
Affinity DataIC50: 1nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as reduction of rise in intracellular Ca2+ concentration after 60 to 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532612(CHEMBL4459054)
Affinity DataIC50: 1nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as blocking of inward/outward currents after 20 to 48 hrs in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532612(CHEMBL4459054)
Affinity DataIC50: 1nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as blocking of inward/outward currents after 20 to 48 hrs in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532609(CHEMBL4466158)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as reduction of rise in intracellular Ca2+ concentration after 60 to 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532609(CHEMBL4466158)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as reduction of rise in intracellular Ca2+ concentration after 60 to 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532608(CHEMBL4525688)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as reduction of rise in intracellular Ca2+ concentration after 60 to 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532608(CHEMBL4525688)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as reduction of rise in intracellular Ca2+ concentration after 60 to 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532610(CHEMBL4451083)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as blocking of inward/outward currents after 20 to 48 hrs in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532610(CHEMBL4451083)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as blocking of inward/outward currents after 20 to 48 hrs in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532611(CHEMBL4562137)
Affinity DataIC50: 8.40nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as blocking of inward/outward currents after 20 to 48 hrs in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532611(CHEMBL4562137)
Affinity DataIC50: 8.40nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as blocking of inward/outward currents after 20 to 48 hrs in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532609(CHEMBL4466158)
Affinity DataIC50: 9nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as blocking of inward/outward currents after 20 to 48 hrs in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532609(CHEMBL4466158)
Affinity DataIC50: 9nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as blocking of inward/outward currents after 20 to 48 hrs in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532613(CHEMBL4464289)
Affinity DataIC50: 23nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as blocking of inward/outward currents after 20 to 48 hrs in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532613(CHEMBL4464289)
Affinity DataIC50: 23nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as blocking of inward/outward currents after 20 to 48 hrs in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532613(CHEMBL4464289)
Affinity DataIC50: 27nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as reduction of rise in intracellular Ca2+ concentration after 60 to 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532613(CHEMBL4464289)
Affinity DataIC50: 27nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as reduction of rise in intracellular Ca2+ concentration after 60 to 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532610(CHEMBL4451083)
Affinity DataIC50: 31nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as reduction of rise in intracellular Ca2+ concentration after 60 to 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532610(CHEMBL4451083)
Affinity DataIC50: 31nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as reduction of rise in intracellular Ca2+ concentration after 60 to 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532611(CHEMBL4562137)
Affinity DataIC50: 100nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as reduction of rise in intracellular Ca2+ concentration after 60 to 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetShort transient receptor potential channel 5(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50532611(CHEMBL4562137)
Affinity DataIC50: 100nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as reduction of rise in intracellular Ca2+ concentration after 60 to 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed