Compile Data Set for Download or QSAR
Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50047776
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189564(CHEMBL3827241)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189641(CHEMBL3827510)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189666(CHEMBL3827617)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189690(CHEMBL3827050)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189691(CHEMBL3828133)
Affinity DataEC50:  1.24E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189692(CHEMBL3827740)
Affinity DataEC50:  4.38E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189693(CHEMBL3826990)
Affinity DataEC50:  2.01E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189694(CHEMBL3827584)
Affinity DataEC50:  4.27E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189559(CHEMBL3827709)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189560(CHEMBL3828201)
Affinity DataEC50:  414nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189561(CHEMBL3828330)
Affinity DataEC50:  2.38E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189562(CHEMBL3828487)
Affinity DataEC50:  2.06E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189563(CHEMBL3827940)
Affinity DataEC50:  8.61E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50: >1.61E+3nMAssay Description:Agonist activity at full length human PPAR-gamma transfected in human HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189565(CHEMBL3827378)
Affinity DataEC50:  2.18E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189566(CHEMBL3827820)
Affinity DataEC50:  2.86E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189567(CHEMBL3828232)
Affinity DataEC50:  9.17E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189575(CHEMBL3827335)
Affinity DataEC50:  2.82E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  4.51E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189641(CHEMBL3827510)
Affinity DataEC50:  6.80nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189666(CHEMBL3827617)
Affinity DataEC50:  5.60nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189690(CHEMBL3827050)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189691(CHEMBL3828133)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189692(CHEMBL3827740)
Affinity DataEC50:  11nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189693(CHEMBL3826990)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189694(CHEMBL3827584)
Affinity DataEC50:  4nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189565(CHEMBL3827378)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human GR by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha/LXR-beta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human LXR by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human PPAR-delta by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM28800(2-{[(3-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  317nMAssay Description:Agonist activity at rat PPAR-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM28800(2-{[(3-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  426nMAssay Description:Agonist activity at mouse PPAR-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189575(CHEMBL3827335)
Affinity DataEC50:  18nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189567(CHEMBL3828232)
Affinity DataEC50:  94nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189566(CHEMBL3827820)
Affinity DataEC50:  8.60nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human RXR by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189564(CHEMBL3827241)
Affinity DataEC50:  15nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189563(CHEMBL3827940)
Affinity DataEC50:  59nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189562(CHEMBL3828487)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189561(CHEMBL3828330)
Affinity DataEC50:  4.30nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189560(CHEMBL3828201)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189559(CHEMBL3827709)
Affinity DataEC50: >2.50E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  123nMAssay Description:Agonist activity at rat PPAR-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  144nMAssay Description:Agonist activity at mouse PPAR-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at full length human PPAR-alpha transfected in human HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM28802(2-{[(5-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-...)
Affinity DataIC50: 97nMAssay Description:Binding affinity to human GST-tagged PPAR-alpha LBD expressed in Escherichia coli BL21 (DE3) PlysS after 30 mins in presence of fluorescein ligand FL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189566(CHEMBL3827820)
Affinity DataIC50: 671nMAssay Description:Binding affinity to human GST-tagged PPAR-alpha LBD expressed in Escherichia coli BL21 (DE3) PlysS after 30 mins in presence of fluorescein ligand FL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189575(CHEMBL3827335)
Affinity DataIC50: 1.34E+3nMAssay Description:Binding affinity to human GST-tagged PPAR-alpha LBD expressed in Escherichia coli BL21 (DE3) PlysS after 30 mins in presence of fluorescein ligand FL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50189567(CHEMBL3828232)
Affinity DataIC50: 1.56E+3nMAssay Description:Binding affinity to human GST-tagged PPAR-alpha LBD expressed in Escherichia coli BL21 (DE3) PlysS after 30 mins in presence of fluorescein ligand FL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
Displayed 1 to 50 (of 66 total ) | Next | Last >>
Jump to: