Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 7565
TargetATP-dependent translocase ABCB1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202570(4-bromo-2-methoxy-N-(2,4,5-trimethoxyphenyl)benzam...)
Affinity DataIC50: 1.54E+3nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202567(2,4,5-Trimethoxy-N-(2-methoxy-phenyl)-benzamide (1...)
Affinity DataIC50: 3.52E+3nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM81939(NSC_62969 | VERAPAMIL | CAS_52-53-9)
Affinity DataIC50: 3.53E+3nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202563(N-(4-Bromo-phenyl)-2,4,5-trimethoxy-benzamide (10))
Affinity DataIC50: 9.27E+3nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202564(N-(4-Bromo-phenyl)-2,3,4-trimethoxy-benzamide (11))
Affinity DataIC50: 1.94E+4nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202560(2,4,5-Trimethoxy-N-phenyl-benzamide (6))
Affinity DataIC50: 2.19E+4nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202566(3,4,5-Trimethoxy-N-(2-methoxy-phenyl)-benzamide (1...)
Affinity DataIC50: 2.62E+4nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM50363079(CHEMBL1944863 | N-(4-bromophenyl)-3,4,5-trimethoxy...)
Affinity DataIC50: 2.70E+4nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202568(2,3,4-Trimethoxy-N-(2-methoxy-phenyl)-benzamide (1...)
Affinity DataIC50: 3.04E+4nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202569(2,4,6-Trimethoxy-N-(2-methoxy-phenyl)-benzamide (1...)
Affinity DataIC50: 4.76E+4nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202559(3,4,5-trimethoxy-N-phenylbenzamide (5))
Affinity DataIC50: 7.07E+4nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202568(2,3,4-Trimethoxy-N-(2-methoxy-phenyl)-benzamide (1...)
Affinity DataIC50: 7.10E+4nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202565(N-(4-Bromo-phenyl)-2,4,6-trimethoxy-benzamide (12))
Affinity DataIC50: 7.62E+4nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202559(3,4,5-trimethoxy-N-phenylbenzamide (5))
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202560(2,4,5-Trimethoxy-N-phenyl-benzamide (6))
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202561(2,3,4-Trimethoxy-N-phenyl-benzamide (7))
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202562(2,4,6-Trimethoxy-N-phenyl-benzamide (8))
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM50363079(CHEMBL1944863 | N-(4-bromophenyl)-3,4,5-trimethoxy...)
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202563(N-(4-Bromo-phenyl)-2,4,5-trimethoxy-benzamide (10))
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202564(N-(4-Bromo-phenyl)-2,3,4-trimethoxy-benzamide (11))
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202565(N-(4-Bromo-phenyl)-2,4,6-trimethoxy-benzamide (12))
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202566(3,4,5-Trimethoxy-N-(2-methoxy-phenyl)-benzamide (1...)
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202567(2,4,5-Trimethoxy-N-(2-methoxy-phenyl)-benzamide (1...)
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202561(2,3,4-Trimethoxy-N-phenyl-benzamide (7))
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202569(2,4,6-Trimethoxy-N-(2-methoxy-phenyl)-benzamide (1...)
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202570(4-bromo-2-methoxy-N-(2,4,5-trimethoxyphenyl)benzam...)
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Universit�� Di Bari Aldo Moro

LigandPNGBDBM202562(2,4,6-Trimethoxy-N-phenyl-benzamide (8))
Affinity DataIC50: 1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details Article
PubMed