Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50047784
TargetAcetylcholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50313079(Mestinon | Regonol | Pyridostigmine | CHEMBL812 | ...)
Affinity DataIC50: 350nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189893(CHEMBL3828679)
Affinity DataIC50: 460nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetCholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189893(CHEMBL3828679)
Affinity DataIC50: 590nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetCholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50313079(Mestinon | Regonol | Pyridostigmine | CHEMBL812 | ...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189894(CHEMBL3827011)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetCholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189894(CHEMBL3827011)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189895(CHEMBL3828028)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetCholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189895(CHEMBL3828028)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189896(CHEMBL3827624)
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189892(CHEMBL3827856)
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189888(CHEMBL3827449)
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189891(CHEMBL3828644)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189887(CHEMBL3827347)
Affinity DataIC50: 2.60E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189889(CHEMBL3828273)
Affinity DataIC50: 2.80E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetCholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189896(CHEMBL3827624)
Affinity DataIC50: 3.10E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetCholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189892(CHEMBL3827856)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetCholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189888(CHEMBL3827449)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189890(CHEMBL3828739)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetCholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189889(CHEMBL3828273)
Affinity DataIC50: 8.00E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetCholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189887(CHEMBL3827347)
Affinity DataIC50: 9.00E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetCholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189891(CHEMBL3828644)
Affinity DataIC50: 1.03E+6nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed
TargetCholinesterase(Human)
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189890(CHEMBL3828739)
Affinity DataIC50: 1.19E+6nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2017
Entry Details Article
PubMed