Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50009921
TargetTrypsin(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533536(CHEMBL4483694)
Affinity DataKi:  0.160nMAssay Description:Inhibition of trypsin (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533535(CHEMBL4440685)
Affinity DataKi:  6.90nMAssay Description:Inhibition of trypsin (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetPlasminogen(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533536(CHEMBL4483694)
Affinity DataKi:  28nMAssay Description:Inhibition of plasmin (unknown origin) using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor XII(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533535(CHEMBL4440685)
Affinity DataKi:  110nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor XII(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533538(CHEMBL4577000)
Affinity DataKi:  180nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetPlasminogen(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533535(CHEMBL4440685)
Affinity DataKi:  270nMAssay Description:Inhibition of plasmin (unknown origin) using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533539(CHEMBL4470708)
Affinity DataKi:  360nMAssay Description:Inhibition of factor 10a (unknown origin) using Ac-QRSRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533535(CHEMBL4440685)
Affinity DataKi:  460nMAssay Description:Inhibition of factor 10a (unknown origin) using Ac-QRSRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor XII(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533537(CHEMBL4590811)
Affinity DataKi:  490nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor XII(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533533(CHEMBL4449980)
Affinity DataKi:  510nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533538(CHEMBL4577000)
Affinity DataKi:  570nMAssay Description:Inhibition of factor 10a (unknown origin) using Ac-QRSRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor XII(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533536(CHEMBL4483694)
Affinity DataKi:  750nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetPlasminogen(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533533(CHEMBL4449980)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of plasmin (unknown origin) using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor XII(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533534(CHEMBL4446504)
Affinity DataKi:  2.16E+3nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533533(CHEMBL4449980)
Affinity DataKi:  2.24E+3nMAssay Description:Inhibition of trypsin (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor XII(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533539(CHEMBL4470708)
Affinity DataKi:  2.39E+3nMAssay Description:Inhibition of factor 12a (unknown origin) using Ac-QRFRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetPlasminogen(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533537(CHEMBL4590811)
Affinity DataKi:  4.54E+3nMAssay Description:Inhibition of plasmin (unknown origin) using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533537(CHEMBL4590811)
Affinity DataKi:  6.24E+3nMAssay Description:Inhibition of trypsin (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533534(CHEMBL4446504)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of thrombin (unknown origin) using Ac-ATPRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533536(CHEMBL4483694)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of thrombin (unknown origin) using Ac-ATPRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetPlasminogen(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533534(CHEMBL4446504)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of plasmin (unknown origin) using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533535(CHEMBL4440685)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of factor 11a (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533536(CHEMBL4483694)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of factor 10a (unknown origin) using Ac-QRSRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533534(CHEMBL4446504)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of trypsin (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533533(CHEMBL4449980)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of uPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533534(CHEMBL4446504)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of uPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533534(CHEMBL4446504)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of tPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533533(CHEMBL4449980)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human plasma kallikrein using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533535(CHEMBL4440685)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human plasma kallikrein using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533533(CHEMBL4449980)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of thrombin (unknown origin) using Ac-ATPRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533533(CHEMBL4449980)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of tPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533536(CHEMBL4483694)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of tPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533536(CHEMBL4483694)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of uPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533535(CHEMBL4440685)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of tPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533536(CHEMBL4483694)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human plasma kallikrein using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533535(CHEMBL4440685)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of thrombin (unknown origin) using Ac-ATPRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533536(CHEMBL4483694)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of factor 11a (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533535(CHEMBL4440685)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of factor 9a (unknown origin) using Ac-QGRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533534(CHEMBL4446504)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of factor 9a (unknown origin) using Ac-QGRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533533(CHEMBL4449980)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of factor 9a (unknown origin) using Ac-QGRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533534(CHEMBL4446504)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of factor 11a (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533536(CHEMBL4483694)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of factor 9a (unknown origin) using Ac-QGRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533535(CHEMBL4440685)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of uPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533534(CHEMBL4446504)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human plasma kallikrein using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533533(CHEMBL4449980)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of factor 11a (unknown origin) using Bz-FVRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProthrombin(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533537(CHEMBL4590811)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of thrombin (unknown origin) using Ac-ATPRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCoagulation factor IX(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533537(CHEMBL4590811)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of factor 9a (unknown origin) using Ac-QGRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533537(CHEMBL4590811)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of uPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533537(CHEMBL4590811)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of tPA (unknown origin) incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50533537(CHEMBL4590811)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human plasma kallikrein using Ac-RM(O2)YRpNA as substrate incubated for 30 mins measured for 7 mins by morrison plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
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