Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50047798
TargetKelch-like ECH-associated protein 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50190617(CHEMBL3827626)
Affinity DataIC50: 100nMAssay Description:Inhibition of human Keap1 kelch domain (Ala321 to Thr609 residues) binding to fluorescent labeled Nrf2 peptide preincubated for 15 mins followed by N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2017
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50190589(CHEMBL3827630)
Affinity DataIC50: 200nMAssay Description:Inhibition of human Keap1 kelch domain (Ala321 to Thr609 residues) binding to fluorescent labeled Nrf2 peptide preincubated for 15 mins followed by N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2017
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50190618(CHEMBL3827019)
Affinity DataIC50: 200nMAssay Description:Inhibition of human Keap1 kelch domain (Ala321 to Thr609 residues) binding to fluorescent labeled Nrf2 peptide preincubated for 15 mins followed by N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2017
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50190586(CHEMBL3827061)
Affinity DataIC50: 400nMAssay Description:Inhibition of human Keap1 kelch domain (Ala321 to Thr609 residues) binding to fluorescent labeled Nrf2 peptide preincubated for 15 mins followed by N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2017
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50190587(CHEMBL3827496)
Affinity DataIC50: 700nMAssay Description:Inhibition of human Keap1 kelch domain (Ala321 to Thr609 residues) binding to fluorescent labeled Nrf2 peptide preincubated for 15 mins followed by N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2017
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50190588(CHEMBL3826983)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of human Keap1 kelch domain (Ala321 to Thr609 residues) binding to fluorescent labeled Nrf2 peptide preincubated for 15 mins followed by N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2017
Entry Details Article
PubMed