Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50048821
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.800nMAssay Description:Half-maximal inhibition of binding of [125I]CCK-8 to Cholecystokinin receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228290(CHEMBL1907959)
Affinity DataIC50: 3nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228291(CHEMBL296718)
Affinity DataIC50: 4nMAssay Description:Half-maximal inhibition of binding of [125I]CCK-8 to Cholecystokinin receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228287(CHEMBL1907960)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228280(CHEMBL47186)
Affinity DataIC50: 7nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50018287(CHEMBL297534 | {3-[(Naphthalene-2-carbonyl)-amino]...)
Affinity DataIC50: 7.5nMAssay Description:Half-maximal inhibition of binding of [125I]CCK-8 to Cholecystokinin receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228283(CHEMBL297816)
Affinity DataIC50: 28nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228284(CHEMBL47296)
Affinity DataIC50: 35nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228297(CHEMBL43769)
Affinity DataIC50: 60nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228298(CHEMBL295524)
Affinity DataIC50: 110nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228288(CHEMBL294980)
Affinity DataIC50: 130nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228289(CHEMBL2093119)
Affinity DataIC50: 200nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228286(CHEMBL412881)
Affinity DataIC50: 200nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228293(CHEMBL45166)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228294(CHEMBL295203)
Affinity DataIC50: 2.10E+3nMAssay Description:Half-maximal inhibition of binding of [125I]CCK-8 to Cholecystokinin receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228285(CHEMBL296734)
Affinity DataIC50: 2.30E+3nMAssay Description:Half-maximal inhibition of binding of [125I]CCK-8 to Cholecystokinin receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228292(CHEMBL44911)
Affinity DataIC50: 2.70E+3nMAssay Description:Half-maximal inhibition of binding of [125I]CCK-8 to Cholecystokinin receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228282(CHEMBL47593)
Affinity DataIC50: 6.80E+3nMAssay Description:Half-maximal inhibition of binding of [125I]CCK-8 to Cholecystokinin receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228296(CHEMBL47535)
Affinity DataIC50: 5.00E+4nMAssay Description:Half-maximal inhibition of binding of [125I]CCK-8 to Cholecystokinin receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228281(CHEMBL295683)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed