Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50001838
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018316(CHEMBL51692 | 2-Butyl-3',4'-dimethoxy-biphenyl-4-c...)
Affinity DataIC50: 4nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018341(CHEMBL53001 | 2-Ethyl-3',4'-dimethoxy-biphenyl-4-c...)
Affinity DataIC50: 4nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018315(CHEMBL430969 | 2-Ethynyl-3',4'-dimethoxy-biphenyl-...)
Affinity DataIC50: 5nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018325(CHEMBL53584 | [1,1';2',1'']Terphenyl-4'-carboxylic...)
Affinity DataIC50: 5nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018321(CHEMBL53585 | 3',4'-Dimethoxy-biphenyl-4-carboxyli...)
Affinity DataIC50: 15nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018338(CHEMBL53867 | 2-Butyl-3',4'-dimethoxy-biphenyl-4-c...)
Affinity DataIC50: 18nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018337(CHEMBL51238 | 3'-Methoxy-biphenyl-4-carboxylic aci...)
Affinity DataIC50: 20nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018320(CHEMBL432324 | 3',4'-Dimethoxy-2-propyl-biphenyl-4...)
Affinity DataIC50: 50nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018324(CHEMBL299760 | [1,1';2',1'']Terphenyl-4'-carboxyli...)
Affinity DataIC50: 50nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018329(CHEMBL54041 | 3',4'-Dimethoxy-biphenyl-4-carbothio...)
Affinity DataIC50: 60nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018326(CHEMBL296169 | 2-Allyl-3',4'-dimethoxy-biphenyl-4-...)
Affinity DataIC50: 80nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018322(CHEMBL50250 | 4,4''-Dimethoxy-[1,1';2',1'']terphen...)
Affinity DataIC50: 125nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018336(CHEMBL300644 | 3',4'-Dimethoxy-biphenyl-4-carbothi...)
Affinity DataIC50: 140nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018327(CHEMBL53750 | 2-Bromo-3',4'-dimethoxy-biphenyl-4-c...)
Affinity DataIC50: 180nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018323(CHEMBL53808 | 3,3''-Dimethoxy-[1,1';2',1'']terphen...)
Affinity DataIC50: 200nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018328(CHEMBL51867 | 3',4'-Dimethyl-biphenyl-4-carboxylic...)
Affinity DataIC50: 200nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018319(CHEMBL53534 | 3',4'-Dimethoxy-2-nitro-biphenyl-4-c...)
Affinity DataIC50: 200nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018331(CHEMBL53482 | 3',4'-Dimethoxy-2-nitro-biphenyl-4-c...)
Affinity DataIC50: 200nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018330(CHEMBL52636 | 2-Bromo-3',4'-dimethoxy-biphenyl-4-c...)
Affinity DataIC50: 220nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018318(CHEMBL412441 | 3'-Methoxy-biphenyl-4-carboxylic ac...)
Affinity DataIC50: 280nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018333(CHEMBL52031 | 2,3',4'-Trimethoxy-biphenyl-4-carbox...)
Affinity DataIC50: 300nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018317(CHEMBL416480 | 3'-Hydroxy-biphenyl-4-carboxylic ac...)
Affinity DataIC50: 300nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018332(CHEMBL51170 | 3',4'-Dimethoxy-biphenyl-4-carboxyli...)
Affinity DataIC50: 400nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018334(CHEMBL54095 | 3'-Methyl-biphenyl-4-carboxylic acid...)
Affinity DataIC50: 500nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018335(CHEMBL416120 | Biphenyl-4-carboxylic acid (4-pyrid...)
Affinity DataIC50: 630nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018339(CHEMBL50050 | 3'-(Cyclohepta-1,3,5-trienyloxy)-bip...)
Affinity DataIC50: 700nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50018340(CHEMBL301388 | 2,3'-Difluoro-biphenyl-4-carboxylic...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed