Compile Data Set for Download or QSAR
Report error Found 138 Enz. Inhib. hit(s) with all data for entry = 50048177
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  0.280nMAssay Description:Agonist activity at CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  1.90nMAssay Description:Agonist activity at CB1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50160434(AM630 | (6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-...)
Affinity DataKi:  31nMAssay Description:Inverse agonist activity at CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  40nMAssay Description:Agonist activity at CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  40nMAssay Description:Agonist activity at CB1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207242(CHEMBL3901140)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207267(CHEMBL3960083)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207259(CHEMBL3892181)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207271(CHEMBL594935)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207256(CHEMBL3898407)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207255(CHEMBL3944807)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207261(CHEMBL3891003)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207239(CHEMBL3907898)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207242(CHEMBL3901140)
Affinity DataIC50: 300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207269(CHEMBL3907434)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207271(CHEMBL594935)
Affinity DataIC50: 400nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207247(CHEMBL3920181)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207254(CHEMBL3938131)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207259(CHEMBL3892181)
Affinity DataIC50: 500nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207255(CHEMBL3944807)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207244(CHEMBL3916891)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207257(CHEMBL3950235)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207266(CHEMBL3932295)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207258(CHEMBL3889952)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207245(CHEMBL3898882)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207263(CHEMBL3922512)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207271(CHEMBL594935)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207240(CHEMBL3917967)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207244(CHEMBL3916891)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207250(CHEMBL3915743)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207267(CHEMBL3960083)
Affinity DataIC50: 700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM106773(2‐(4‐methoxyphenyl)‐1‐[(4&...)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207255(CHEMBL3944807)
Affinity DataIC50: 800nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207241(CHEMBL3895577)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207262(CHEMBL3898880)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207258(CHEMBL3889952)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207258(CHEMBL3889952)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207251(CHEMBL3916164)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207256(CHEMBL3898407)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207271(CHEMBL594935)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207244(CHEMBL3916891)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207261(CHEMBL3891003)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207239(CHEMBL3907898)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207255(CHEMBL3944807)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207265(CHEMBL3914550)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207269(CHEMBL3907434)
Affinity DataIC50: 1.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207270(CHEMBL3926929)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207252(CHEMBL3935866)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207248(CHEMBL3904520)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Pontificia Universidad Cat£Lica De Chile

Curated by ChEMBL
LigandPNGBDBM50207247(CHEMBL3920181)
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2018
Entry Details Article
PubMed
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