Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50047909
TargetGlycogen phosphorylase, liver form(Human)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50065965(5-Chloro-1H-indole-2-carboxylic acid [2-((R)-dimet...)
Affinity DataIC50: 82nMAssay Description:Inhibition of human recombinant liver glycogen phosphorylase A expressed in baculovirus infected Sf9 insect cells assessed as release of phosphate fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196903(CHEMBL3916767)
Affinity DataIC50: 178nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b using 10 mM of glucose-1-phosphate as substrate preincubated for 60 mins followed by substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196903(CHEMBL3916767)
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant liver glycogen phosphorylase A expressed in baculovirus infected Sf9 insect cells assessed as release of phosphate fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50263771(N-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymet...)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50295859((2S,3R,4R,5S,6R)-2-(1H-benzo[d]imidazol-2-yl)-6-(h...)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as inorganic phosphate release using glucose-1-phosphate as substrate by doubl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50295859((2S,3R,4R,5S,6R)-2-(1H-benzo[d]imidazol-2-yl)-6-(h...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b using alpha-D-glucose-1-phosphate as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen phosphorylase, liver form(Human)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196901(CHEMBL3986514)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human recombinant liver glycogen phosphorylase A expressed in baculovirus infected Sf9 insect cells assessed as release of phosphate fr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50295860((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...)
Affinity DataKi:  7.60E+4nMAssay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as inorganic phosphate release using glucose-1-phosphate as substrate by doubl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50295860((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...)
Affinity DataKi:  2.29E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b using alpha-D-glucose-1-phosphate as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196912(CHEMBL3969601)
Affinity DataIC50: 3.24E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196904(CHEMBL3952333)
Affinity DataIC50: 3.58E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196909(CHEMBL3915666)
Affinity DataIC50: 3.97E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196911(CHEMBL3932944)
Affinity DataIC50: 4.02E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196908(CHEMBL3897672)
Affinity DataIC50: 4.37E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196906(CHEMBL3925760)
Affinity DataIC50: 5.08E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196905(CHEMBL3906675)
Affinity DataIC50: 5.16E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196910(CHEMBL3943625)
Affinity DataIC50: 5.31E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196907(CHEMBL3904951)
Affinity DataIC50: 5.32E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50196902(CHEMBL3931874)
Affinity DataIC50: 6.22E+5nMpH: 6.8Assay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as reduction in inorganic phosphate release using glucose-1-phosphate as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed