Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50047834
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192837(CHEMBL3964816 | US10188627, Compound 8d)
Affinity DataEC50:  1.60nMAssay Description:Transactivation of ProLink tagged human PPARdelta transfected in CHO-K1 cells assessed as interaction with EA labelled SRCP after 3 to 16 hrs by beta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192832(CHEMBL3975891 | US10188627, Compound 8c)
Affinity DataEC50:  1.90nMAssay Description:Transactivation of ProLink tagged human PPARdelta transfected in CHO-K1 cells assessed as interaction with EA labelled SRCP after 3 to 16 hrs by beta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192829(CHEMBL3958704 | US10188627, Compound 8a)
Affinity DataEC50:  5.10nMAssay Description:Transactivation of ProLink tagged human PPARdelta transfected in CHO-K1 cells assessed as interaction with EA labelled SRCP after 3 to 16 hrs by beta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192830(CHEMBL3983906 | US10188627, Compound 8g)
Affinity DataEC50:  5.5nMAssay Description:Transactivation of ProLink tagged human PPARdelta transfected in CHO-K1 cells assessed as interaction with EA labelled SRCP after 3 to 16 hrs by beta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192837(CHEMBL3964816 | US10188627, Compound 8d)
Affinity DataEC50:  7.40nMAssay Description:Transactivation of human Gal4-PPARdelta LBD transfected in African green monkey CV1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192836(CHEMBL3911672 | US10188627, Compound 8m)
Affinity DataEC50:  13nMAssay Description:Transactivation of ProLink tagged human PPARdelta transfected in CHO-K1 cells assessed as interaction with EA labelled SRCP after 3 to 16 hrs by beta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192832(CHEMBL3975891 | US10188627, Compound 8c)
Affinity DataEC50:  15nMAssay Description:Transactivation of human Gal4-PPARdelta LBD transfected in African green monkey CV1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192834(CHEMBL3914092 | US10188627, Compound 8n)
Affinity DataEC50:  20nMAssay Description:Transactivation of human Gal4-PPARdelta LBD transfected in African green monkey CV1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192834(CHEMBL3914092 | US10188627, Compound 8n)
Affinity DataEC50:  23nMAssay Description:Transactivation of ProLink tagged human PPARdelta transfected in CHO-K1 cells assessed as interaction with EA labelled SRCP after 3 to 16 hrs by beta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192830(CHEMBL3983906 | US10188627, Compound 8g)
Affinity DataEC50:  40nMAssay Description:Transactivation of human Gal4-PPARdelta LBD transfected in African green monkey CV1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192831(CHEMBL3895104 | US10188627, Compound 8h)
Affinity DataEC50:  40nMAssay Description:Transactivation of ProLink tagged human PPARdelta transfected in CHO-K1 cells assessed as interaction with EA labelled SRCP after 3 to 16 hrs by beta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192829(CHEMBL3958704 | US10188627, Compound 8a)
Affinity DataEC50:  56nMAssay Description:Transactivation of human Gal4-PPARdelta LBD transfected in African green monkey CV1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192833(CHEMBL3923083 | US10188627, Compound 8j)
Affinity DataEC50:  65nMAssay Description:Transactivation of ProLink tagged human PPARdelta transfected in CHO-K1 cells assessed as interaction with EA labelled SRCP after 3 to 16 hrs by beta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192835(CHEMBL3981654 | US10188627, Compound 8x)
Affinity DataEC50:  83nMAssay Description:Transactivation of human Gal4-PPARdelta LBD transfected in African green monkey CV1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192835(CHEMBL3981654 | US10188627, Compound 8x)
Affinity DataEC50:  265nMAssay Description:Transactivation of ProLink tagged human PPARdelta transfected in CHO-K1 cells assessed as interaction with EA labelled SRCP after 3 to 16 hrs by beta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192833(CHEMBL3923083 | US10188627, Compound 8j)
Affinity DataEC50:  566nMAssay Description:Transactivation of human Gal4-PPARdelta LBD transfected in African green monkey CV1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192831(CHEMBL3895104 | US10188627, Compound 8h)
Affinity DataEC50:  998nMAssay Description:Transactivation of human Gal4-PPARdelta LBD transfected in African green monkey CV1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50192836(CHEMBL3911672 | US10188627, Compound 8m)
Affinity DataEC50:  1.32E+3nMAssay Description:Transactivation of human Gal4-PPARdelta LBD transfected in African green monkey CV1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2018
Entry Details Article
PubMed