Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50047959
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198670(CHEMBL3960590)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198661(CHEMBL3955849)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198660(CHEMBL3928231)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198677(CHEMBL3929427)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198662(CHEMBL3966957)
Affinity DataIC50: 56nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198682(CHEMBL3918835)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198678(CHEMBL3891045)
Affinity DataIC50: 140nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198667(CHEMBL3963507)
Affinity DataIC50: 140nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198681(CHEMBL3966515)
Affinity DataIC50: 150nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198680(CHEMBL3983437)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198660(CHEMBL3928231)
Affinity DataIC50: 160nMAssay Description:Displacement of [1,2,6,7-3H]progesterone from recombinant human GST-tagged PR-LBD (675 to 933 residues) expressed in baculovirus-infected insect cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198675(CHEMBL3957000)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198674(CHEMBL3965979)
Affinity DataIC50: 190nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198664(CHEMBL3954803)
Affinity DataIC50: 210nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198657(CHEMBL3960113)
Affinity DataIC50: 220nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198676(CHEMBL3936738)
Affinity DataIC50: 230nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198655(CHEMBL3948334)
Affinity DataIC50: 230nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198668(CHEMBL3955372)
Affinity DataIC50: 240nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198654(CHEMBL3927761)
Affinity DataIC50: 250nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198669(CHEMBL3938469)
Affinity DataIC50: 260nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198656(CHEMBL3946113)
Affinity DataIC50: 290nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198665(CHEMBL3894599)
Affinity DataIC50: 290nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198673(CHEMBL3975572)
Affinity DataIC50: 300nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198659(CHEMBL3946665)
Affinity DataIC50: 340nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198666(CHEMBL3975017)
Affinity DataIC50: 440nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198663(CHEMBL3975442)
Affinity DataIC50: 450nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198671(CHEMBL3924332)
Affinity DataIC50: 480nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355216(CHEMBL1835807)
Affinity DataIC50: 500nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198684(CHEMBL3920525)
Affinity DataIC50: 550nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198672(CHEMBL3939561)
Affinity DataIC50: 570nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198683(CHEMBL3974043)
Affinity DataIC50: 580nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198662(CHEMBL3966957)
Affinity DataIC50: 790nMAssay Description:Displacement of [1,2,6,7-3H]progesterone from recombinant human GST-tagged PR-LBD (675 to 933 residues) expressed in baculovirus-infected insect cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198658(CHEMBL3903073)
Affinity DataIC50: 850nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198670(CHEMBL3960590)
Affinity DataIC50: 990nMAssay Description:Displacement of [1,2,6,7-3H]progesterone from recombinant human GST-tagged PR-LBD (675 to 933 residues) expressed in baculovirus-infected insect cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198668(CHEMBL3955372)
Affinity DataIC50: 1.36E+3nMAssay Description:Displacement of [1,2,6,7-3H]progesterone from recombinant human GST-tagged PR-LBD (675 to 933 residues) expressed in baculovirus-infected insect cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355216(CHEMBL1835807)
Affinity DataIC50: 1.42E+3nMAssay Description:Displacement of [1,2,6,7-3H]progesterone from recombinant human GST-tagged PR-LBD (675 to 933 residues) expressed in baculovirus-infected insect cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355216(CHEMBL1835807)
Affinity DataIC50: 3.54E+3nMAssay Description:Displacement of [3H]dexamethasone from human GR measured after 18 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355216(CHEMBL1835807)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human ARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198668(CHEMBL3955372)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]dexamethasone from human GR measured after 18 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50355243(CHEMBL1835836)
Affinity DataIC50: 1.52E+4nMAssay Description:Displacement of [1,2,6,7-3H]progesterone from recombinant human GST-tagged PR-LBD (675 to 933 residues) expressed in baculovirus-infected insect cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198673(CHEMBL3975572)
Affinity DataIC50: 1.57E+4nMAssay Description:Displacement of [1,2,6,7-3H]progesterone from recombinant human GST-tagged PR-LBD (675 to 933 residues) expressed in baculovirus-infected insect cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50198679(CHEMBL3937217)
Affinity DataIC50: 1.58E+4nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase expression after 24 hrs by alkaline...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed