Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50000705
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50249298(N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimethylcarbami...)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259113(CHEMBL4090253)
Affinity DataIC50: 21nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259086(CHEMBL4076970)
Affinity DataIC50: 42nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259075(CHEMBL4063484)
Affinity DataIC50: 127nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259110(CHEMBL4062243)
Affinity DataIC50: 157nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259115(CHEMBL4059479)
Affinity DataIC50: 165nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259076(CHEMBL4071434)
Affinity DataIC50: 234nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259109(CHEMBL4082407)
Affinity DataIC50: 345nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259118(CHEMBL4100421)
Affinity DataIC50: 498nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259116(CHEMBL4066602)
Affinity DataIC50: 532nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259119(CHEMBL4070862)
Affinity DataIC50: 717nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259079(CHEMBL4067693)
Affinity DataIC50: 887nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259078(CHEMBL4093380)
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259077(CHEMBL4097741)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259074(CHEMBL4081450)
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259114(CHEMBL4097963)
Affinity DataIC50: 2.21E+3nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259080(CHEMBL4089030)
Affinity DataIC50: 4.07E+3nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetProthrombin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50249298(N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimethylcarbami...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human thrombin using substrate S-2238 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate rea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259081(CHEMBL4084611)
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetProthrombin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259113(CHEMBL4090253)
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of human thrombin using substrate S-2238 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate rea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetProthrombin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259086(CHEMBL4076970)
Affinity DataIC50: 8.10E+4nMAssay Description:Inhibition of human thrombin using substrate S-2238 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate rea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259084(CHEMBL4091746)
Affinity DataIC50: 1.13E+5nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259083(CHEMBL4102953)
Affinity DataIC50: 1.79E+5nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259082(CHEMBL4062061)
Affinity DataIC50: 2.43E+5nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259117(CHEMBL4090100)
Affinity DataIC50: 3.54E+5nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50259085(CHEMBL4065217)
Affinity DataIC50: 5.46E+5nMAssay Description:Inhibition of human factor 10a using substrate S-2765 preincubated for 30 mins followed by substrate addition measured after 20 mins by micro plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2019
Entry Details Article
PubMed