Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50048265
TargetAlpha-1D adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50419716(CHEMBL1946777)
Affinity DataKi:  0.813nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1d adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210789(CHEMBL3938383)
Affinity DataKi:  0.933nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HeLa cell membranes after 30 mins by TopCount liquid scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50026917(CHEMBL13647 | BMY 7378 | 8-{2-[4-(2-Methoxy-phenyl...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HeLa cell membranes after 30 mins by TopCount liquid scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50026917(CHEMBL13647 | BMY 7378 | 8-{2-[4-(2-Methoxy-phenyl...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1d adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210792(CHEMBL3917316)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HeLa cell membranes after 30 mins by TopCount liquid scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210791(CHEMBL3901382)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HeLa cell membranes after 30 mins by TopCount liquid scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210795(CHEMBL3929328)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HeLa cell membranes after 30 mins by TopCount liquid scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210790(CHEMBL3981480)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HeLa cell membranes after 30 mins by TopCount liquid scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210794(CHEMBL3892434)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HeLa cell membranes after 30 mins by TopCount liquid scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50099434(CHEMBL2234448)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HeLa cell membranes after 30 mins by TopCount liquid scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50419716(CHEMBL1946777)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HeLa cell membranes after 30 mins by TopCount liquid scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210796(CHEMBL3970754)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HeLa cell membranes after 30 mins by TopCount liquid scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210791(CHEMBL3901382)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1d adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210789(CHEMBL3938383)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1d adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210793(CHEMBL1183249)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HeLa cell membranes after 30 mins by TopCount liquid scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210794(CHEMBL3892434)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1d adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210794(CHEMBL3892434)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1a adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50099434(CHEMBL2234448)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1a adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210790(CHEMBL3981480)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1d adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210795(CHEMBL3929328)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1d adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210792(CHEMBL3917316)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1d adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50099434(CHEMBL2234448)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1b adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210789(CHEMBL3938383)
Affinity DataKi:  186nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1a adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210794(CHEMBL3892434)
Affinity DataKi:  191nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1b adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210789(CHEMBL3938383)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1b adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210795(CHEMBL3929328)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1a adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210796(CHEMBL3970754)
Affinity DataKi:  214nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1d adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210791(CHEMBL3901382)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1b adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210790(CHEMBL3981480)
Affinity DataKi:  229nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1a adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210791(CHEMBL3901382)
Affinity DataKi:  269nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1a adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210790(CHEMBL3981480)
Affinity DataKi:  389nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1b adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50026917(CHEMBL13647 | BMY 7378 | 8-{2-[4-(2-Methoxy-phenyl...)
Affinity DataKi:  389nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1a adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210795(CHEMBL3929328)
Affinity DataKi:  407nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1b adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210796(CHEMBL3970754)
Affinity DataKi:  437nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1b adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210793(CHEMBL1183249)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1d adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210792(CHEMBL3917316)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1b adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50026917(CHEMBL13647 | BMY 7378 | 8-{2-[4-(2-Methoxy-phenyl...)
Affinity DataKi:  708nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1b adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210793(CHEMBL1183249)
Affinity DataKi:  977nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1b adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210792(CHEMBL3917316)
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1a adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210788(CHEMBL3911497)
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1a adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50099434(CHEMBL2234448)
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1d adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210796(CHEMBL3970754)
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1a adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210788(CHEMBL3911497)
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HeLa cell membranes after 30 mins by TopCount liquid scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210793(CHEMBL1183249)
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1a adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210788(CHEMBL3911497)
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1b adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50210788(CHEMBL3911497)
Affinity DataKi:  1.78E+3nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha1d adrenergic receptor expressed in CHO cell membranes after 30 mins by TopCount liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed