Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50001864
TargetThromboxane A2 receptor(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50228336(CHEMBL71879)
Affinity DataIC50: 2.10nMAssay Description:In vitro concentration that reduced specific binding of [3H]U-440619 to guinea pig platelet receptor, TXA2 by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50279755(7-Phenyl-7-(2,4,5-trimethyl-3,6-dioxo-cyclohexa-1,...)
Affinity DataIC50: 7.40nMAssay Description:In vitro concentration that reduced specific binding of [3H]U-440619 to guinea pig platelet receptor, TXA2 by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50292409((Z)-7-((1R,4S,5S,6R)-6-((S,E)-3-hydroxyoct-1-enyl)...)
Affinity DataIC50: 31nMAssay Description:In vitro concentration that reduced specific binding of [3H]U-440619 to guinea pig platelet receptor, Thromboxane A2 receptor by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetThromboxane A2 receptor(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50228337(CHEMBL71921)
Affinity DataIC50: 210nMAssay Description:In vitro concentration that reduced specific binding of [3H]U-440619 to guinea pig platelet receptor, TXA2 by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed