Compile Data Set for Download or QSAR
Report error Found 102 Enz. Inhib. hit(s) with all data for entry = 50000719
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259594(CHEMBL4068321)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259630(CHEMBL4079843)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259595(CHEMBL4097867)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259597(CHEMBL4105601)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259593(CHEMBL4095676)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM76662(7-Benzyloxy-4-methyl-chromen-2-one | 4-methyl-7-ph...)
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259629(CHEMBL4094745)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259631(CHEMBL4082300)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50378564(CHEMBL145781)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 7nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition measured after 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259604(CHEMBL4060398)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 17nMAssay Description:Inhibition of equine serum BuChE using S-butylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259606(CHEMBL4069084)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259597(CHEMBL4105601)
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259595(CHEMBL4097867)
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259605(CHEMBL4090150)
Affinity DataIC50: 73nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 102nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition measured after 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259603(CHEMBL4087723)
Affinity DataIC50: 104nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259594(CHEMBL4068321)
Affinity DataIC50: 240nMAssay Description:Inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259633(CHEMBL4067432)
Affinity DataIC50: 290nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259624(CHEMBL4088674)
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259630(CHEMBL4079843)
Affinity DataIC50: 370nMAssay Description:Inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259622(CHEMBL4078343)
Affinity DataIC50: 470nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259623(CHEMBL4096387)
Affinity DataIC50: 530nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259631(CHEMBL4082300)
Affinity DataIC50: 600nMAssay Description:Inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259606(CHEMBL4069084)
Affinity DataIC50: 720nMAssay Description:Inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259629(CHEMBL4094745)
Affinity DataIC50: 960nMAssay Description:Inhibition of equine serum BuChE using S-butylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259604(CHEMBL4060398)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259633(CHEMBL4067432)
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of equine serum BuChE using S-butylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259593(CHEMBL4095676)
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259628(CHEMBL4089608)
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259627(CHEMBL4104128)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259634(CHEMBL4066437)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259629(CHEMBL4094745)
Affinity DataIC50: 2.13E+3nMAssay Description:Inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM76662(7-Benzyloxy-4-methyl-chromen-2-one | 4-methyl-7-ph...)
Affinity DataIC50: 2.62E+3nMAssay Description:Inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 2.87E+3nMAssay Description:Inhibition of equine serum BuChE using S-butylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259617(CHEMBL4091054)
Affinity DataIC50: 3.09E+3nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259627(CHEMBL4104128)
Affinity DataIC50: 3.12E+3nMAssay Description:Inhibition of equine serum BuChE using S-butylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50378564(CHEMBL145781)
Affinity DataIC50: 3.49E+3nMAssay Description:Inhibition of recombinant human MAO-A assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259626(CHEMBL4086218)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259623(CHEMBL4096387)
Affinity DataIC50: 5.19E+3nMAssay Description:Inhibition of equine serum BuChE using S-butylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259625(CHEMBL4093982)
Affinity DataIC50: 5.33E+3nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259640(CHEMBL4061479)
Affinity DataIC50: 5.64E+3nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259624(CHEMBL4088674)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of equine serum BuChE using S-butylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259624(CHEMBL4088674)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition measured after 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259632(CHEMBL4063174)
Affinity DataIC50: 9.21E+3nMAssay Description:Inhibition of recombinant human MAO-B assessed as reduction in 4-hydroxyquinolone production using kynuramine as substrate after 20 mins by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM76662(7-Benzyloxy-4-methyl-chromen-2-one | 4-methyl-7-ph...)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of equine serum BuChE using S-butylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of The Western Cape

Curated by ChEMBL
LigandPNGBDBM50259626(CHEMBL4086218)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of equine serum BuChE using S-butylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition measured after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2020
Entry Details Article
PubMed
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