Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50011230
TargetBromodomain-containing protein 1(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  1.65E+3nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: E556-A688More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetTranscription intermediary factor 1-alpha(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  8.48E+3nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: G861-E979More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetTranscription initiation factor TFIID subunit 1-like(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  2.50E+4nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: M1401-D1522More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetTranscription initiation factor TFIID subunit 1(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  17nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: D1522-D1656More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetTranscription initiation factor TFIID subunit 1(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  5.53E+3nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: R1398-D1524More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  1.97E+4nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: L1451-E1580More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  4.76E+3nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: G715-D831More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetProtein polybromo-1(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  1.42E+4nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: S613-D734More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  1.89E+3nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: S2791-H2911More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetChromatin remodeling regulator CECR2(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  8nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: P420-D543More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetBromodomain and PHD finger-containing protein 3(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  8.62E+3nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: L591-P711More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  172nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: S257-E382More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  40nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: N21-E137More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  50nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: E348-D455More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2A(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  3.75E+3nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: H1769-Q1872More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetChromatin remodeling regulator CECR2(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataIC50: 9.40nMAssay Description:Alphascreen assay. Binding to CECR2A (domain start/stop: P420-H538) by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetBromodomain-containing protein 9(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataIC50: 47nMAssay Description:Homogeneous Time Resolved Fluorescence (HTRF) assay. Domain start/stop: L14-Q143More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetChromatin remodeling regulator CECR2(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataIC50: 48nMAssay Description:Alphascreen assay. Binding to CECR2A (domain start/stop: P420-D543) by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetChromatin remodeling regulator CECR2(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataIC50: 79nMAssay Description:Alphascreen assay. Binding to CECR2A (domain start/stop: P420-D543) by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataIC50: 83nMAssay Description:Alphascreen assay. Binding to BRD4A (domain start/stop: N44-E168) by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataIC50: 116nMAssay Description:Homogeneous Time Resolved Fluorescence (HTRF) assay. Domain start/stop: N44-E168More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetPeregrin(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataIC50: 141nMAssay Description:Alphascreen assay. Binding to BRPF1B (domain start/stop: M626-G740) by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetBromodomain-containing protein 9(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataIC50: 300nMAssay Description:Alphascreen assay. Binding to BRD9A (domain start/stop: L14-Q143) by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataIC50: 311nMAssay Description:Alphascreen assay. Binding to BRD4A (domain start/stop: N44-E168) by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataIC50: 468nMAssay Description:Alphascreen assay. Binding to BRD4A (domain start/stop: N44-E168) by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetBromodomain-containing protein 9(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataIC50: 701nMAssay Description:Alphascreen assay. Binding to BRD9A (domain start/stop: L14-Q143) by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataIC50: 2.44E+3nMAssay Description:Alphascreen assay. Binding to CREBBPA (domain start/stop: R1081-G1197) by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed