Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50048184
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207359(CHEMBL3892377)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207351(CHEMBL3965256)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207353(CHEMBL3949755)
Affinity DataIC50: 0.670nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207349(CHEMBL3958414)
Affinity DataIC50: 0.840nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207350(CHEMBL3956954)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207353(CHEMBL3949755)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207355(CHEMBL3987106)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50318884(CHEMBL1084546 | CHEMBL2430359 | N-methyl-N-(3-((2-...)
Affinity DataIC50: 1.5nMAssay Description:Reversible/competitive inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207365(CHEMBL3899046)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207356(CHEMBL3969464)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207352(CHEMBL3908093)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207354(CHEMBL3961368)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207362(CHEMBL3977870)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207361(CHEMBL3889951)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207350(CHEMBL3956954)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207355(CHEMBL3987106)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207364(CHEMBL3936048)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207348(CHEMBL3912281)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207349(CHEMBL3958414)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207356(CHEMBL3969464)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207365(CHEMBL3899046)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207352(CHEMBL3908093)
Affinity DataIC50: 9.20nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207354(CHEMBL3961368)
Affinity DataIC50: 10nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207348(CHEMBL3912281)
Affinity DataIC50: 11nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50318884(CHEMBL1084546 | CHEMBL2430359 | N-methyl-N-(3-((2-...)
Affinity DataIC50: 13nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207362(CHEMBL3977870)
Affinity DataIC50: 14nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207361(CHEMBL3889951)
Affinity DataIC50: 17nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207351(CHEMBL3965256)
Affinity DataIC50: 20nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207357(CHEMBL3939286)
Affinity DataIC50: 21nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207357(CHEMBL3939286)
Affinity DataIC50: 26nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207358(CHEMBL3914036)
Affinity DataIC50: 27nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207358(CHEMBL3914036)
Affinity DataIC50: 30nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207359(CHEMBL3892377)
Affinity DataIC50: 122nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207360(CHEMBL3927099)
Affinity DataIC50: 177nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207360(CHEMBL3927099)
Affinity DataIC50: 201nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207364(CHEMBL3936048)
Affinity DataIC50: 256nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetProtein-tyrosine kinase 2-beta(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207363(CHEMBL3898282)
Affinity DataIC50: 6.63E+3nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged PYK2 expressed in baculovirus infected sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50207363(CHEMBL3898282)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed