Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50048166
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206900(CHEMBL3895181)
Affinity DataIC50: 0.0300nMAssay Description:Antagonist activity at GR in human HepG2 cells assessed as inhibition of protein mediated-transcriptional activity by MMTV-promoter driven luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206899(CHEMBL3964460)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at GR in human HepG2 cells assessed as protein mediated-transcriptional activity by MMTV-promoter driven luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206940(CHEMBL3981243)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at GR in human HepG2 cells assessed as protein mediated-transcriptional activity by MMTV-promoter driven luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206950(CHEMBL3933702)
Affinity DataIC50: 0.0700nMAssay Description:Antagonist activity at GR in human HepG2 cells assessed as inhibition of protein mediated-transcriptional activity by MMTV-promoter driven luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206900(CHEMBL3895181)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at GR in human HepG2 cells assessed as protein mediated-transcriptional activity by MMTV-promoter driven luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206947(CHEMBL3966490)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at GR in human HepG2 cells assessed as inhibition of protein mediated-transcriptional activity by MMTV-promoter driven luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206952(CHEMBL3907029)
Affinity DataIC50: 0.900nMAssay Description:Antagonist activity at GR in human HepG2 cells assessed as inhibition of protein mediated-transcriptional activity by MMTV-promoter driven luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206951(CHEMBL3904106)
Affinity DataIC50: 1.40nMAssay Description:Antagonist activity at GR in human HepG2 cells assessed as inhibition of protein mediated-transcriptional activity by MMTV-promoter driven luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206944(CHEMBL3927299)
Affinity DataIC50: 37nMAssay Description:Antagonist activity at GR in human HepG2 cells assessed as inhibition of protein mediated-transcriptional activity by MMTV-promoter driven luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206945(CHEMBL3909248)
Affinity DataEC50:  47nMAssay Description:Agonist activity at GR in human HepG2 cells assessed as protein mediated-transcriptional activity by MMTV-promoter driven luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206953(CHEMBL3982975)
Affinity DataIC50: 84nMAssay Description:Antagonist activity at GR in human HepG2 cells assessed as inhibition of protein mediated-transcriptional activity by MMTV-promoter driven luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206935(CHEMBL3956011)
Affinity DataIC50: 91nMAssay Description:Antagonist activity at GR in human HepG2 cells assessed as inhibition of protein mediated-transcriptional activity by MMTV-promoter driven luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206934(CHEMBL3937005)
Affinity DataEC50:  100nMAssay Description:Agonist activity at GR in human HepG2 cells assessed as protein mediated-transcriptional activity by MMTV-promoter driven luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206949(CHEMBL3891049)
Affinity DataEC50:  149nMAssay Description:Agonist activity at GR in human HepG2 cells assessed as protein mediated-transcriptional activity by MMTV-promoter driven luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206902(CHEMBL3983602)
Affinity DataEC50:  240nMAssay Description:Agonist activity at GR in human HepG2 cells assessed as protein mediated-transcriptional activity by MMTV-promoter driven luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206954(CHEMBL3937406)
Affinity DataEC50:  265nMAssay Description:Agonist activity at GR in human HepG2 cells assessed as protein mediated-transcriptional activity by MMTV-promoter driven luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206946(CHEMBL3954977)
Affinity DataEC50:  280nMAssay Description:Agonist activity at GR in human HepG2 cells assessed as protein mediated-transcriptional activity by MMTV-promoter driven luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206898(CHEMBL3967119)
Affinity DataIC50: 455nMAssay Description:Antagonist activity at GR in human HepG2 cells assessed as inhibition of protein mediated-transcriptional activity by MMTV-promoter driven luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206903(CHEMBL3928010)
Affinity DataIC50: 558nMAssay Description:Antagonist activity at GR in human HepG2 cells assessed as inhibition of protein mediated-transcriptional activity by MMTV-promoter driven luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206954(CHEMBL3937406)
Affinity DataIC50: 626nMAssay Description:Antagonist activity at GR in human HepG2 cells assessed as inhibition of protein mediated-transcriptional activity by MMTV-promoter driven luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206949(CHEMBL3891049)
Affinity DataIC50: 1.36E+3nMAssay Description:Antagonist activity at GR in human HepG2 cells assessed as inhibition of protein mediated-transcriptional activity by MMTV-promoter driven luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206901(CHEMBL3894105)
Affinity DataEC50:  1.86E+3nMAssay Description:Agonist activity at GR in human HepG2 cells assessed as protein mediated-transcriptional activity by MMTV-promoter driven luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206934(CHEMBL3937005)
Affinity DataIC50: 2.35E+3nMAssay Description:Antagonist activity at GR in human HepG2 cells assessed as inhibition of protein mediated-transcriptional activity by MMTV-promoter driven luciferase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50206944(CHEMBL3927299)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at GR in human HepG2 cells assessed as protein mediated-transcriptional activity by MMTV-promoter driven luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed