Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50012612
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558761(CHEMBL4783674)
Affinity DataEC50:  690nMAssay Description:Agonist activity at human delta opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558761(CHEMBL4783674)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human kappa opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50170678(CHEMBL363324 | (3S,4aR,4bS,6S,8R,8aR,10aR)-6-Benzo...)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human kappa opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50189145((2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 9-acetoxy-2-(f...)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human kappa opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558762(CHEMBL4749616)
Affinity DataEC50:  0.560nMAssay Description:Agonist activity at human kappa opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50159165(2S,4aR,6a(R,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human kappa opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataEC50:  780nMAssay Description:Agonist activity at human delta opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558750(CHEMBL4790712)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human delta opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558751(CHEMBL4745430)
Affinity DataEC50:  620nMAssay Description:Agonist activity at human delta opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558752(CHEMBL4760942)
Affinity DataEC50:  770nMAssay Description:Agonist activity at human delta opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558753(CHEMBL4741711)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human delta opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558754(CHEMBL4799292)
Affinity DataEC50:  310nMAssay Description:Agonist activity at human delta opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558755(CHEMBL4756271)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human delta opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558756(CHEMBL4782368)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human delta opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558757(CHEMBL4763725)
Affinity DataEC50:  180nMAssay Description:Agonist activity at human delta opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558759(CHEMBL4786506)
Affinity DataEC50:  74nMAssay Description:Agonist activity at human delta opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558760(CHEMBL4752988)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human kappa opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50170678(CHEMBL363324 | (3S,4aR,4bS,6S,8R,8aR,10aR)-6-Benzo...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human delta opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50159165(2S,4aR,6a(R,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human delta opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment measured after 90 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment measured after 90 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558750(CHEMBL4790712)
Affinity DataEC50:  96nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment measured after 90 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558751(CHEMBL4745430)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment measured after 90 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558752(CHEMBL4760942)
Affinity DataEC50:  330nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment measured after 90 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558753(CHEMBL4741711)
Affinity DataEC50:  360nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment measured after 90 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558754(CHEMBL4799292)
Affinity DataEC50:  180nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment measured after 90 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558755(CHEMBL4756271)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment measured after 90 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558756(CHEMBL4782368)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment measured after 90 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558757(CHEMBL4763725)
Affinity DataEC50:  63nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment measured after 90 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558759(CHEMBL4786506)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment measured after 90 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558761(CHEMBL4783674)
Affinity DataEC50:  560nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment measured after 90 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50170678(CHEMBL363324 | (3S,4aR,4bS,6S,8R,8aR,10aR)-6-Benzo...)
Affinity DataEC50:  3.40E+3nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment measured after 90 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50189145((2S,4aR,6aR,7R,9R,10aS,10bR)-methyl 9-acetoxy-2-(f...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558750(CHEMBL4790712)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558751(CHEMBL4745430)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558752(CHEMBL4760942)
Affinity DataEC50:  31nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558753(CHEMBL4741711)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558754(CHEMBL4799292)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558755(CHEMBL4756271)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558756(CHEMBL4782368)
Affinity DataEC50:  4.70nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558757(CHEMBL4763725)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50265928(CHEMBL4086641)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558758(CHEMBL4787274)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558759(CHEMBL4786506)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558760(CHEMBL4752988)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558761(CHEMBL4783674)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50170678(CHEMBL363324 | (3S,4aR,4bS,6S,8R,8aR,10aR)-6-Benzo...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50558762(CHEMBL4749616)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human mu opiod receptor expressed in CHO-K1 cells assessed as increase in forskolin induced cAMP production measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
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