Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 7808
TargetPlasma kallikrein(Human)
University of Glasgow

LigandPNGBDBM218837(TBMB-PK15 (10))
Affinity DataKi:  1.30nMpH: 7.4Assay Description:The inhibition of plasma kallikrein and coagulation factor FXII was assessed by incubating the proteases with bicyclic peptide (twofold dilutions) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2017
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
University of Glasgow

LigandPNGBDBM218839(TBMT-FX618 (16) | TBMT-PK15 (12))
Affinity DataKi:  20nMpH: 7.4Assay Description:The inhibition of plasma kallikrein and coagulation factor FXII was assessed by incubating the proteases with bicyclic peptide (twofold dilutions) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2017
Entry Details Article
PubMed
TargetCoagulation factor XII(Human)
University of Glasgow

LigandPNGBDBM218840(TATA-FXII618 (14))
Affinity DataKi:  25nMpH: 7.4Assay Description:The inhibition of plasma kallikrein and coagulation factor FXII was assessed by incubating the proteases with bicyclic peptide (twofold dilutions) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2017
Entry Details Article
PubMed
TargetCoagulation factor XII(Human)
University of Glasgow

LigandPNGBDBM218838(TATB-FXII618 (15) | TATB-PK15 (11))
Affinity DataKi:  340nMpH: 7.4Assay Description:The inhibition of plasma kallikrein and coagulation factor FXII was assessed by incubating the proteases with bicyclic peptide (twofold dilutions) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2017
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
University of Glasgow

LigandPNGBDBM218838(TATB-FXII618 (15) | TATB-PK15 (11))
Affinity DataKi:  540nMpH: 7.4Assay Description:The inhibition of plasma kallikrein and coagulation factor FXII was assessed by incubating the proteases with bicyclic peptide (twofold dilutions) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2017
Entry Details Article
PubMed
TargetCoagulation factor XII(Human)
University of Glasgow

LigandPNGBDBM218839(TBMT-FX618 (16) | TBMT-PK15 (12))
Affinity DataKi:  1.22E+3nMpH: 7.4Assay Description:The inhibition of plasma kallikrein and coagulation factor FXII was assessed by incubating the proteases with bicyclic peptide (twofold dilutions) an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2017
Entry Details Article
PubMed