Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50048057
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203146(CHEMBL3902533)
Affinity DataIC50: 0.996nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203125(CHEMBL3917936)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203124(CHEMBL3916619)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203118(CHEMBL3962242)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203114(CHEMBL3936937)
Affinity DataIC50: 5nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203116(CHEMBL3925782)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203117(CHEMBL3934673)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203152(CHEMBL3964039)
Affinity DataIC50: 8.80nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203150(CHEMBL3980079)
Affinity DataIC50: 10nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203115(CHEMBL3986381)
Affinity DataIC50: 14nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203151(CHEMBL3962160)
Affinity DataIC50: 14nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203149(CHEMBL3954524)
Affinity DataIC50: 16nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203148(CHEMBL3909003)
Affinity DataIC50: 24nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203120(CHEMBL3927938)
Affinity DataIC50: 118nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203119(CHEMBL3899948)
Affinity DataIC50: 634nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203147(CHEMBL3893222)
Affinity DataIC50: 687nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203123(CHEMBL3926893)
Affinity DataIC50: 734nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50203121(CHEMBL3945821)
Affinity DataIC50: 757nMAssay Description:Inhibition of human activated ERK2 assessed as reduction in phosphorylation activity preincubated for 15 mins followed by addition of IMAP peptide as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed