Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50049088
TargetTryptophan 5-hydroxylase 2(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50233990(CHEMBL4104957)
Affinity DataIC50: 7nMAssay Description:Inhibition of TPH2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234204(CHEMBL4077986)
Affinity DataIC50: 11nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234218(CHEMBL4086156)
Affinity DataIC50: 14nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234203(CHEMBL4064649)
Affinity DataIC50: 19nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50233988(CHEMBL4097252)
Affinity DataIC50: 20nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234202(CHEMBL4072840)
Affinity DataIC50: 21nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50233987(CHEMBL4084634)
Affinity DataIC50: 22nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234217(CHEMBL4104549)
Affinity DataIC50: 22nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234201(CHEMBL4078797)
Affinity DataIC50: 23nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234211(CHEMBL4079227)
Affinity DataIC50: 23nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234205(CHEMBL4088856)
Affinity DataIC50: 25nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234206(CHEMBL4060885)
Affinity DataIC50: 26nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234200(CHEMBL4094630)
Affinity DataIC50: 26nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145634(CHEMBL3764999)
Affinity DataIC50: 26nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234219(CHEMBL4095779)
Affinity DataIC50: 28nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234199(CHEMBL4063143)
Affinity DataIC50: 30nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234216(CHEMBL4090304)
Affinity DataIC50: 30nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234207(CHEMBL4065816)
Affinity DataIC50: 30nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50233986(CHEMBL4092679)
Affinity DataIC50: 32nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234198(CHEMBL4105500)
Affinity DataIC50: 32nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234208(CHEMBL4093347)
Affinity DataIC50: 32nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50233990(CHEMBL4104957)
Affinity DataIC50: 33nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234002(CHEMBL4072764)
Affinity DataIC50: 35nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234103(CHEMBL4085937)
Affinity DataIC50: 35nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234209(CHEMBL4065734)
Affinity DataIC50: 37nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234220(CHEMBL4077881)
Affinity DataIC50: 39nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234215(CHEMBL4071484)
Affinity DataIC50: 40nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234210(CHEMBL4074348)
Affinity DataIC50: 40nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234001(CHEMBL4073070)
Affinity DataIC50: 51nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234214(CHEMBL4084194)
Affinity DataIC50: 53nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50233998(CHEMBL4099936)
Affinity DataIC50: 53nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50233997(CHEMBL4061688)
Affinity DataIC50: 62nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50233995(CHEMBL4091280)
Affinity DataIC50: 65nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50233994(CHEMBL4076761)
Affinity DataIC50: 73nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234213(CHEMBL4061818)
Affinity DataIC50: 77nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50233993(CHEMBL4084339)
Affinity DataIC50: 207nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50233991(CHEMBL4060643)
Affinity DataIC50: 460nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50233992(CHEMBL4074718)
Affinity DataIC50: 885nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed
TargetTryptophan 5-hydroxylase 1(Human)
Karos Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50234212(CHEMBL4065512)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of TPH1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2019
Entry Details Article
PubMed