Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with all data for entry = 50000741
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50203424(CHEMBL3893393)
Affinity DataIC50: 0.158nMAssay Description:Transrepression activity at glucocorticoid receptor in human THP1 cells assessed as receptor-mediated anti-inflammatory activity by measuring inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50203424(CHEMBL3893393)
Affinity DataIC50: 0.158nMAssay Description:Transrepression activity at glucocorticoid receptorin human HeLa cells assessed as inhibition of TPA-induced collagenase promoter activity by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50203424(CHEMBL3893393)
Affinity DataIC50: 0.631nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM18207(dexamethasone (tetramethyl-rhodamine conjugated ) ...)
Affinity DataIC50: 1.60nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM18207(dexamethasone (tetramethyl-rhodamine conjugated ) ...)
Affinity DataIC50: 2.5nMAssay Description:Transrepression activity at glucocorticoid receptor in human THP1 cells assessed as receptor-mediated anti-inflammatory activity by measuring inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259977(CHEMBL4082878)
Affinity DataIC50: 2.5nMAssay Description:Binding affinity to recombinant human glucocorticoid receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259977(CHEMBL4082878)
Affinity DataIC50: 4nMAssay Description:Transrepression activity at glucocorticoid receptorin human HeLa cells assessed as inhibition of TPA-induced collagenase promoter activity by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259977(CHEMBL4082878)
Affinity DataIC50: 4nMAssay Description:Transrepression activity at glucocorticoid receptor in human THP1 cells assessed as receptor-mediated anti-inflammatory activity by measuring inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50416869(CHEMBL1257572)
Affinity DataIC50: 5nMAssay Description:Transrepression activity at glucocorticoid receptor in human THP1 cells assessed as receptor-mediated anti-inflammatory activity by measuring inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50416869(CHEMBL1257572)
Affinity DataIC50: 5nMAssay Description:Transrepression activity at glucocorticoid receptorin human HeLa cells assessed as inhibition of TPA-induced collagenase promoter activity by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259978(CHEMBL4069357)
Affinity DataIC50: 5nMAssay Description:Transrepression activity at glucocorticoid receptor in human THP1 cells assessed as receptor-mediated anti-inflammatory activity by measuring inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259978(CHEMBL4069357)
Affinity DataIC50: 5nMAssay Description:Transrepression activity at glucocorticoid receptorin human HeLa cells assessed as inhibition of TPA-induced collagenase promoter activity by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50416869(CHEMBL1257572)
Affinity DataIC50: 5.01nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259979(CHEMBL4090392)
Affinity DataIC50: 6.30nMAssay Description:Transrepression activity at glucocorticoid receptor in human THP1 cells assessed as receptor-mediated anti-inflammatory activity by measuring inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259981(CHEMBL4085241)
Affinity DataIC50: 6.30nMAssay Description:Transrepression activity at glucocorticoid receptorin human HeLa cells assessed as inhibition of TPA-induced collagenase promoter activity by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50203426(CHEMBL3962413)
Affinity DataIC50: 6.30nMAssay Description:Transrepression activity at glucocorticoid receptorin human HeLa cells assessed as inhibition of TPA-induced collagenase promoter activity by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50416869(CHEMBL1257572)
Affinity DataIC50: 6.30nMAssay Description:Binding affinity to recombinant human glucocorticoid receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259981(CHEMBL4085241)
Affinity DataIC50: 6.30nMAssay Description:Transrepression activity at glucocorticoid receptor in human THP1 cells assessed as receptor-mediated anti-inflammatory activity by measuring inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259979(CHEMBL4090392)
Affinity DataIC50: 6.30nMAssay Description:Transrepression activity at glucocorticoid receptorin human HeLa cells assessed as inhibition of TPA-induced collagenase promoter activity by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50203426(CHEMBL3962413)
Affinity DataIC50: 6.30nMAssay Description:Transrepression activity at glucocorticoid receptor in human THP1 cells assessed as receptor-mediated anti-inflammatory activity by measuring inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM18207(dexamethasone (tetramethyl-rhodamine conjugated ) ...)
Affinity DataIC50: 7.90nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50203426(CHEMBL3962413)
Affinity DataIC50: 10nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM18207(dexamethasone (tetramethyl-rhodamine conjugated ) ...)
Affinity DataIC50: 13nMAssay Description:Binding affinity to recombinant human glucocorticoid receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259978(CHEMBL4069357)
Affinity DataIC50: 13nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259981(CHEMBL4085241)
Affinity DataIC50: 13nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259978(CHEMBL4069357)
Affinity DataIC50: 13nMAssay Description:Binding affinity to recombinant human glucocorticoid receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259980(CHEMBL4092066)
Affinity DataIC50: 16nMAssay Description:Transrepression activity at glucocorticoid receptorin human HeLa cells assessed as inhibition of TPA-induced collagenase promoter activity by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259980(CHEMBL4092066)
Affinity DataIC50: 16nMAssay Description:Transrepression activity at glucocorticoid receptor in human THP1 cells assessed as receptor-mediated anti-inflammatory activity by measuring inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259980(CHEMBL4092066)
Affinity DataIC50: 16nMAssay Description:Binding affinity to recombinant human glucocorticoid receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259986(CHEMBL4098118)
Affinity DataIC50: 16nMAssay Description:Binding affinity to recombinant human glucocorticoid receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259984(CHEMBL4072079)
Affinity DataIC50: 20nMAssay Description:Transrepression activity at glucocorticoid receptor in human THP1 cells assessed as receptor-mediated anti-inflammatory activity by measuring inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259984(CHEMBL4072079)
Affinity DataIC50: 20nMAssay Description:Transrepression activity at glucocorticoid receptorin human HeLa cells assessed as inhibition of TPA-induced collagenase promoter activity by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259986(CHEMBL4098118)
Affinity DataIC50: 20nMAssay Description:Transrepression activity at glucocorticoid receptor in human THP1 cells assessed as receptor-mediated anti-inflammatory activity by measuring inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259986(CHEMBL4098118)
Affinity DataIC50: 20nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259981(CHEMBL4085241)
Affinity DataIC50: 20nMAssay Description:Binding affinity to recombinant human glucocorticoid receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259977(CHEMBL4082878)
Affinity DataIC50: 25nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259980(CHEMBL4092066)
Affinity DataIC50: 25nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259979(CHEMBL4090392)
Affinity DataIC50: 25nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50203424(CHEMBL3893393)
Affinity DataIC50: 32nMAssay Description:Binding affinity to recombinant human glucocorticoid receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259986(CHEMBL4098118)
Affinity DataIC50: 40nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259985(CHEMBL4064352)
Affinity DataIC50: 40nMAssay Description:Transrepression activity at glucocorticoid receptor in human THP1 cells assessed as receptor-mediated anti-inflammatory activity by measuring inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259985(CHEMBL4064352)
Affinity DataIC50: 40nMAssay Description:Transrepression activity at glucocorticoid receptorin human HeLa cells assessed as inhibition of TPA-induced collagenase promoter activity by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50203426(CHEMBL3962413)
Affinity DataIC50: 63nMAssay Description:Binding affinity to recombinant human glucocorticoid receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259984(CHEMBL4072079)
Affinity DataIC50: 63nMAssay Description:Binding affinity to recombinant human glucocorticoid receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259985(CHEMBL4064352)
Affinity DataIC50: 126nMAssay Description:Binding affinity to recombinant human glucocorticoid receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259979(CHEMBL4090392)
Affinity DataIC50: 126nMAssay Description:Binding affinity to recombinant human glucocorticoid receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259984(CHEMBL4072079)
Affinity DataIC50: 158nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259985(CHEMBL4064352)
Affinity DataIC50: 158nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259977(CHEMBL4082878)
Affinity DataIC50: 200nMAssay Description:Binding affinity to recombinant human progesterone receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259981(CHEMBL4085241)
Affinity DataIC50: 316nMAssay Description:Binding affinity to recombinant human androgen receptor expressed in baculovirus infected sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2020
Entry Details Article
PubMed
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