Compile Data Set for Download or QSAR
Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 50049137
LigandPNGBDBM50235076(CHEMBL4073137)
Affinity DataEC50:  339nMAssay Description:Inhibition of NET (unknown origin) expressed in HEK293 cells assessed as reduction in norepinephrine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235078(CHEMBL4092912)
Affinity DataEC50:  5.20nMAssay Description:Agonist activity at human beta3 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235122(CHEMBL4065251)
Affinity DataEC50:  5.10nMAssay Description:Agonist activity at human beta3 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235077(CHEMBL4074920)
Affinity DataEC50:  251nMAssay Description:Inhibition of NET (unknown origin) expressed in HEK293 cells assessed as reduction in norepinephrine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235119(CHEMBL4085173)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human beta3 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235079(CHEMBL4103112)
Affinity DataEC50:  827nMAssay Description:Inhibition of NET (unknown origin) expressed in HEK293 cells assessed as reduction in norepinephrine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235122(CHEMBL4065251)
Affinity DataEC50:  1.52E+3nMAssay Description:Inhibition of NET (unknown origin) expressed in HEK293 cells assessed as reduction in norepinephrine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235121(CHEMBL4066314)
Affinity DataEC50:  65nMAssay Description:Inhibition of NET (unknown origin) expressed in HEK293 cells assessed as reduction in norepinephrine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235121(CHEMBL4066314)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human beta3 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235120(CHEMBL4087670)
Affinity DataEC50:  26nMAssay Description:Inhibition of NET (unknown origin) expressed in HEK293 cells assessed as reduction in norepinephrine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235120(CHEMBL4087670)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at human beta3 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235075(CHEMBL4095361)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at human beta3 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235119(CHEMBL4085173)
Affinity DataEC50:  627nMAssay Description:Inhibition of NET (unknown origin) expressed in HEK293 cells assessed as reduction in norepinephrine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235079(CHEMBL4103112)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at human beta3 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235078(CHEMBL4092912)
Affinity DataEC50:  1.39E+3nMAssay Description:Inhibition of NET (unknown origin) expressed in HEK293 cells assessed as reduction in norepinephrine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235077(CHEMBL4074920)
Affinity DataEC50:  0.320nMAssay Description:Agonist activity at human beta3 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235075(CHEMBL4095361)
Affinity DataEC50:  254nMAssay Description:Inhibition of NET (unknown origin) expressed in HEK293 cells assessed as reduction in norepinephrine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235076(CHEMBL4073137)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human beta3 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235077(CHEMBL4074920)
Affinity DataIC50: 8.79E+3nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235119(CHEMBL4085173)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235120(CHEMBL4087670)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235075(CHEMBL4095361)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235122(CHEMBL4065251)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235076(CHEMBL4073137)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235079(CHEMBL4103112)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235078(CHEMBL4092912)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235121(CHEMBL4066314)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235076(CHEMBL4073137)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235121(CHEMBL4066314)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235075(CHEMBL4095361)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235078(CHEMBL4092912)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235122(CHEMBL4065251)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235122(CHEMBL4065251)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235121(CHEMBL4066314)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235076(CHEMBL4073137)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235120(CHEMBL4087670)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235120(CHEMBL4087670)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235079(CHEMBL4103112)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235079(CHEMBL4103112)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235119(CHEMBL4085173)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235119(CHEMBL4085173)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235078(CHEMBL4092912)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235077(CHEMBL4074920)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235075(CHEMBL4095361)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50235077(CHEMBL4074920)
Affinity DataIC50: 2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235119(CHEMBL4085173)
Affinity DataIC50: 2.99E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235122(CHEMBL4065251)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.5 by electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235075(CHEMBL4095361)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.5 by electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235077(CHEMBL4074920)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.5 by electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
LigandPNGBDBM50235119(CHEMBL4085173)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.5 by electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
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