Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50048248
TargetEstrogen receptor(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 0.410nMAssay Description:Displacement of fluormone-labeled ES2 from recombinant full length human ERalpha ligand binding domain expressed in insect cells after 2 hrs by TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50180684(4-OHT | Afimoxifene | TamoGel)
Affinity DataIC50: 0.530nMAssay Description:Displacement of fluormone-labeled ES2 from recombinant full length human ERalpha ligand binding domain expressed in insect cells after 2 hrs by TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50210071(CHEMBL3885342)
Affinity DataIC50: 1.10nMAssay Description:Displacement of fluormone-labeled ES2 from recombinant full length human ERalpha ligand binding domain expressed in insect cells after 2 hrs by TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50090463(CHEMBL3581633)
Affinity DataIC50: 14nMAssay Description:Displacement of fluormone-labeled ES2 from recombinant full length human ERalpha ligand binding domain expressed in insect cells after 2 hrs by TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50210071(CHEMBL3885342)
Affinity DataIC50: 210nMAssay Description:Downregulation of ERalpha in human MCF7 cells after 4 hrs by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50090463(CHEMBL3581633)
Affinity DataIC50: 220nMAssay Description:Downregulation of ERalpha in human MCF7 cells after 4 hrs by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed