Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50048287
TargetPeroxisome proliferator-activated receptor gamma(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50030474(US9562012, rosiglitazone | CHEBI:50122 | Avandamet...)
Affinity DataIC50: 292nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211660(CHEMBL3915254)
Affinity DataIC50: 350nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211669(CHEMBL3943220)
Affinity DataIC50: 369nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211676(CHEMBL3899514)
Affinity DataIC50: 482nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211656(CHEMBL3959627)
Affinity DataIC50: 491nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211677(CHEMBL3977442)
Affinity DataIC50: 1.14E+3nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211659(CHEMBL3949291)
Affinity DataIC50: 1.15E+3nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211658(CHEMBL3986626)
Affinity DataIC50: 1.29E+3nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211657(CHEMBL3941555)
Affinity DataIC50: 1.32E+3nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2018
Entry Details Article
PubMed