Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 7786
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM217379(CDDO-Me, 2)
Affinity DataIC50: 6.00E+3nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM217380(CDDO-EA, 3)
Affinity DataIC50: 8.00E+3nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM217384(Steroid scaffold, 9)
Affinity DataIC50: 8.00E+3nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM80086(cid_9958995 | (4aR,6aR,6aS,6bR,8aS,12aS,14bS)-8a-i...)
Affinity DataIC50: 3.80E+4nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM217381(CDDO-TFEA, 4)
Affinity DataIC50: 4.40E+4nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM217385(Steroid scaffold, 10)
Affinity DataIC50: 8.30E+4nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM217383(Oleanic acid, 7)
Affinity DataIC50: 1.00E+5nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM50242128(taraxerol | CHEMBL511822 | Taraxerol, 8)
Affinity DataIC50: 1.00E+5nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM217382(Ursolic acid, 6)
Affinity DataIC50: 1.00E+5nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM50096348(2-Cyano-3,12-Dioxooleana-1,9(11)-Dien-28-Oic Acid ...)
Affinity DataIC50: 1.00E+5nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM217386(Steroid scaffold, 11)
Affinity DataIC50: 1.70E+5nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM217387(Steroid scaffold, 12)
Affinity DataIC50: 4.00E+5nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM217388(Steroid scaffold, 13)
Affinity DataIC50: 4.00E+5nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM217390(2-Bromo-2-cyclohexenone, 17)
Affinity DataIC50: 5.00E+5nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM92505(4-Cholesten-3-one | Steroid scaffold, 14)
Affinity DataIC50: 1.00E+6nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM17289(folliculin | (1S,10R,11S,15S)-5-hydroxy-15-methylt...)
Affinity DataIC50: 1.00E+6nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM217389(2-Cyano-2-cyclohexenone, 16)
Affinity DataIC50: 1.20E+6nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed
TargetGhrelin O-acyltransferase(Human)
Syracuse University

LigandPNGBDBM217391(Cyclohexenone, 18)
Affinity DataIC50: 1.00E+6nMpH: 7.0 T: 2°CAssay Description:Assays were performed with ~100 μg of membrane protein, as determined by a Bradford assay. The membrane fraction was preincubated with 1 μM met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2017
Entry Details Article
PubMed