Compile Data Set for Download or QSAR
Report error Found 78 Enz. Inhib. hit(s) with all data for entry = 50049322
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239006(CHEMBL4060481)
Affinity DataIC50: 29nMAssay Description:Inhibition of DRAK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDeath-associated protein kinase 1(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239006(CHEMBL4060481)
Affinity DataKd:  54nMAssay Description:Binding affinity to DAPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239006(CHEMBL4060481)
Affinity DataKd:  99nMAssay Description:Binding affinity to DRAK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238990(CHEMBL4105195)
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238997(CHEMBL4076100)
Affinity DataIC50: 410nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 510nMAssay Description:Inhibition of human TEKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238996(CHEMBL4099371)
Affinity DataIC50: 690nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetAurora kinase A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 850nMAssay Description:Inhibition of human AURORA-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 950nMAssay Description:Inhibition of human TEKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238998(CHEMBL4103220)
Affinity DataIC50: 960nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238995(CHEMBL4072438)
Affinity DataIC50: 990nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetAurora kinase A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human AURORA-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238999(CHEMBL4072264)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239011(CHEMBL4074827)
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50024284(CHEMBL3334979)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238990(CHEMBL4105195)
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of human DRAK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human CDK5More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50024284(CHEMBL3334979)
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of human DRAK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibition of human ITKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 2.16E+3nMAssay Description:Inhibition of human CDK9More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of human ITKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDeath-associated protein kinase 3(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 2.33E+3nMAssay Description:Inhibition of human DAPK3More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239003(CHEMBL4101141)
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of human CDK6More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 2.82E+3nMAssay Description:Inhibition of human CDK4More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase Blk(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 2.88E+3nMAssay Description:Inhibition of human BLKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase Blk(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 3.05E+3nMAssay Description:Inhibition of human BLKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDeath-associated protein kinase 2(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 3.07E+3nMAssay Description:Inhibition of human DAPK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50036932(CHEMBL1478023 | US11866416, Compound SN-II-118)
Affinity DataIC50: 3.08E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238984(CHEMBL2253274)
Affinity DataIC50: 3.11E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238986(CHEMBL2253275)
Affinity DataIC50: 3.24E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239009(CHEMBL4073831)
Affinity DataIC50: 3.66E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 4.26E+3nMAssay Description:Inhibition of human JAK3More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 4.63E+3nMAssay Description:Inhibition of human SYKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238990(CHEMBL4105195)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human BTKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238990(CHEMBL4105195)
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 5.03E+3nMAssay Description:Inhibition of human BTKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase Blk(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238990(CHEMBL4105195)
Affinity DataIC50: 5.26E+3nMAssay Description:Inhibition of human BLKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human GSK3betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239013(CHEMBL4101308)
Affinity DataIC50: 5.37E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 5.81E+3nMAssay Description:Inhibition of human DRAK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17A(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 5.85E+3nMAssay Description:Inhibition of human DRAK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50580(MLS000863576 | (2Z)-2-[(3,4-dihydroxyphenyl)methyl...)
Affinity DataIC50: 6.02E+3nMAssay Description:Inhibition of human BTKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238990(CHEMBL4105195)
Affinity DataIC50: 6.23E+3nMAssay Description:Inhibition of human IKKBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDeath-associated protein kinase 2(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238989(CHEMBL4087337)
Affinity DataIC50: 6.34E+3nMAssay Description:Inhibition of human DAPK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50238985(CHEMBL4093574)
Affinity DataIC50: 6.65E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17B(Human)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50239002(CHEMBL4105654)
Affinity DataIC50: 7.16E+3nMAssay Description:Inhibition of recombinant GST-tagged DRAK2 (unknown origin) autophosphorylation after 2 hrs by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
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