Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50002117
TargetMu-type opioid receptor(Rat)
The First Hospital of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50453766(CHEMBL4210361)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in Wistar rat brain membranes preincubated for 1 hr measured after 1hr by scintillation counting m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The First Hospital of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50453765(CHEMBL4215224)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in Wistar rat brain membranes preincubated for 1 hr measured after 1hr by scintillation counting m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The First Hospital of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in Wistar rat brain membranes preincubated for 1 hr measured after 1hr by scintillation counting m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The First Hospital of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50453764(CHEMBL4211768)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in Wistar rat brain membranes preincubated for 1 hr measured after 1hr by scintillation counting m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
The First Hospital of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50453767(CHEMBL4202727)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in Wistar rat brain membranes preincubated for 1 hr measured after 1hr by scintillation counting m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
The First Hospital of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50453765(CHEMBL4215224)
Affinity DataKi:  2.03E+3nMAssay Description:Displacement of [3H]-DPDPE from delta opioid receptor in Wistar rat brain membranes preincubated for 3 hrs measured after 1 hr by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
The First Hospital of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50453766(CHEMBL4210361)
Affinity DataKi:  3.87E+3nMAssay Description:Displacement of [3H]-DPDPE from delta opioid receptor in Wistar rat brain membranes preincubated for 3 hrs measured after 1 hr by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
The First Hospital of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50453767(CHEMBL4202727)
Affinity DataKi:  4.05E+3nMAssay Description:Displacement of [3H]-DPDPE from delta opioid receptor in Wistar rat brain membranes preincubated for 3 hrs measured after 1 hr by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
The First Hospital of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50453764(CHEMBL4211768)
Affinity DataKi:  4.06E+3nMAssay Description:Displacement of [3H]-DPDPE from delta opioid receptor in Wistar rat brain membranes preincubated for 3 hrs measured after 1 hr by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
The First Hospital of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  5.09E+3nMAssay Description:Displacement of [3H]-DPDPE from delta opioid receptor in Wistar rat brain membranes preincubated for 3 hrs measured after 1 hr by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed