Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50000389
TargetProtein-arginine deiminase type-2(Mouse)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248829(CHEMBL4084229)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of full length recombinant mouse N-terminal GST-tagged PAD2 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethyl ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2019
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248829(CHEMBL4084229)
Affinity DataKi:  4.70E+4nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged PAD4 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethylester ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2019
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-2(Mouse)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataKi:  1.79E+5nMAssay Description:Inhibition of full length recombinant mouse N-terminal GST-tagged PAD2 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethyl ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2019
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataKi:  1.83E+5nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged PAD4 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethylester ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2019
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-1(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248829(CHEMBL4084229)
Affinity DataKi:  3.84E+5nMAssay Description:Inhibition of human PAD1 using BAEE as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2019
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-1(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50426302(CHEMBL2312698)
Affinity DataKi:  4.45E+5nMAssay Description:Inhibition of human PAD1 using BAEE as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2019
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-1(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248824(CHEMBL4059499)
Affinity DataKi:  6.02E+5nMAssay Description:Inhibition of human PAD1 using BAEE as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2019
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248830(CHEMBL4089583)
Affinity DataKi:  6.32E+5nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged PAD4 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethylester ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2019
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-2(Mouse)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248832(CHEMBL4084379)
Affinity DataKi:  7.14E+5nMAssay Description:Inhibition of full length recombinant mouse N-terminal GST-tagged PAD2 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethyl ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2019
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248824(CHEMBL4059499)
Affinity DataKi:  1.43E+6nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged PAD4 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethylester ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2019
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-1(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248814(CHEMBL4070114)
Affinity DataKi:  2.42E+6nMAssay Description:Inhibition of human PAD1 using BAEE as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2019
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-2(Mouse)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248830(CHEMBL4089583)
Affinity DataKi:  4.62E+6nMAssay Description:Inhibition of full length recombinant mouse N-terminal GST-tagged PAD2 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethyl ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2019
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50248831(CHEMBL4102346)
Affinity DataKi:  4.64E+6nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged PAD4 expressed in baculovirus infected Sf9 cells using benzoyl arginine ethylester ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2019
Entry Details Article
PubMed