Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50000950
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159502(CHEMBL3786849)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]OSIP339391 from human recombinant adenosine A2B receptor expressed in HEK293 cell membranes after 60 mins by liquid scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21190(CHEMBL113142 | 4-(2-{[5-amino-2-(furan-2-yl)-[1,2,...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]4-(2-[7-amino-2-(2-furyl)[1,2,4]triazolo[2,3-a][1,3,5]triazin-5-ylamino]ethyl)phenol from human adenosine A2A receptor expressed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50086170(CHEMBL1628266 | N-(4-Cyano-phenyl)-2-[4-(2,6-dioxo...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]ZM241385/[125I]IABOPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50265851(CHEMBL4071734)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50265857(CHEMBL4061502)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159479(CHEMBL1566489)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159480(CHEMBL1544856)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159491(CHEMBL1490082)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50265858(CHEMBL4075899)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50042209(4-(2,6-dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159233(CHEMBL3091704)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50265855(CHEMBL4099777)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21190(CHEMBL113142 | 4-(2-{[5-amino-2-(furan-2-yl)-[1,2,...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50265856(CHEMBL4072891)
Affinity DataKi:  102nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  157nMAssay Description:Displacement of [3H]4-(2-[7-amino-2-(2-furyl)[1,2,4]triazolo[2,3-a][1,3,5]triazin-5-ylamino]ethyl)phenol from human adenosine A2A receptor expressed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50265854(CHEMBL4092030)
Affinity DataKi:  349nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50265853(CHEMBL4079899)
Affinity DataKi:  461nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159489(CHEMBL1606497)
Affinity DataKi:  586nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50265852(CHEMBL4104142)
Affinity DataKi:  647nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21190(CHEMBL113142 | 4-(2-{[5-amino-2-(furan-2-yl)-[1,2,...)
Affinity DataKi:  683nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21190(CHEMBL113142 | 4-(2-{[5-amino-2-(furan-2-yl)-[1,2,...)
Affinity DataKi:  863nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human Hela cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50265859(CHEMBL4083334)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50159483(CHEMBL3091699)
Affinity DataKi:  1.49E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  1.72E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human Hela cell membranes after 180 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed