Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50001942
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM83449(cid_9795678 | PHENCYCLIDINE | SMR001338811 | Phenc...)
Affinity DataKi:  60nMAssay Description:Binding affinity against phencyclidine receptor was determined by the displacement of [3H]TCP of whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50018933(CHEMBL44566 | 1-(3-Methyl-1-phenyl-cyclohexyl)-pip...)
Affinity DataKi:  170nMAssay Description:Binding affinity against phencyclidine receptor was determined by the displacement of [3H]TCP of whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM83449(cid_9795678 | PHENCYCLIDINE | SMR001338811 | Phenc...)
Affinity DataIC50: 600nMAssay Description:Inhibition activity against binding of phencyclidine receptor was determined by the displacement of [3H]-TCP of whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50018932(CHEMBL40424 | 1-(3-Methyl-1-phenyl-cyclohexyl)-pip...)
Affinity DataKi:  820nMAssay Description:Binding affinity against phencyclidine receptor was determined by the displacement of [3H]TCP of whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50018929(CHEMBL42842 | 3-Methyl-1-(1-phenyl-cyclohexyl)-pip...)
Affinity DataKi:  2.15E+3nMAssay Description:Binding affinity against phencyclidine receptor was determined by the displacement of [3H]TCP of whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50018929(CHEMBL42842 | 3-Methyl-1-(1-phenyl-cyclohexyl)-pip...)
Affinity DataKi:  2.15E+3nMAssay Description:Binding affinity against phencyclidine receptor was determined by the displacement of [3H]TCP of whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50018931(CHEMBL288469 | 1-(3-Methyl-1-phenyl-cyclohexyl)-pi...)
Affinity DataKi:  3.30E+3nMAssay Description:Binding affinity against phencyclidine receptor was determined by the displacement of [3H]TCP of whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2C(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50018930(CHEMBL42033 | 1-(3-Methyl-1-phenyl-cyclohexyl)-pip...)
Affinity DataKi:  6.80E+3nMAssay Description:Binding affinity against phencyclidine receptor was determined by the displacement of [3H]TCP of whole rat brain minus cerebellum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed