Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 4869
TargetBeta-arrestin-1(Rabbit)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82381(L-659,989, (-))
Affinity DataKi:  0.510nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829(L-662,418 | (2S,5S)-2-(3-Methanesulfonyl-5-methoxy...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2011
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82381(L-659,989, (-))
Affinity DataKi:  5.48nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829(L-662,418 | (2S,5S)-2-(3-Methanesulfonyl-5-methoxy...)
Affinity DataKi:  12.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2011
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829(L-662,418 | (2S,5S)-2-(3-Methanesulfonyl-5-methoxy...)
Affinity DataKi:  14.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2011
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)
Affinity DataKi:  79.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2011
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829(L-662,418 | (2S,5S)-2-(3-Methanesulfonyl-5-methoxy...)
Affinity DataKi:  152nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829(L-662,418 | (2S,5S)-2-(3-Methanesulfonyl-5-methoxy...)
Affinity DataKi:  205nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2011
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829(L-662,418 | (2S,5S)-2-(3-Methanesulfonyl-5-methoxy...)
Affinity DataKi:  1.11E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2011
Entry Details
PubMed