Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 50049000
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232666(CHEMBL4083059)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-LSD from 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50048803(5-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-et...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-Raclopride from D2L receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232674(CHEMBL4068850)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-LSD from 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232673(CHEMBL4061189)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-LSD from 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM35254(CHEMBL715 | 2-methyl-4-(4-methylpiperazin-1-yl)-10...)
Affinity DataKi:  6.20nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM35254(CHEMBL715 | 2-methyl-4-(4-methylpiperazin-1-yl)-10...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-LSD from 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232672(CHEMBL4090862)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-LSD from 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232667(CHEMBL4060194)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]-LSD from 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232670(CHEMBL4088416)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]-LSD from 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]-5-CT from 5-HT7b receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232671(CHEMBL4096141)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]-LSD from 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232673(CHEMBL4061189)
Affinity DataKi:  65nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232669(CHEMBL4079631)
Affinity DataKi:  266nMAssay Description:Displacement of [3H]-LSD from 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232666(CHEMBL4083059)
Affinity DataKi:  438nMAssay Description:Displacement of [3H]-5-CT from 5-HT7b receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232666(CHEMBL4083059)
Affinity DataKi:  489nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232668(CHEMBL4103891)
Affinity DataKi:  755nMAssay Description:Displacement of [3H]-LSD from 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232666(CHEMBL4083059)
Affinity DataKi:  1.49E+3nMAssay Description:Displacement of [3H]-Raclopride from D2L receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232667(CHEMBL4060194)
Affinity DataKi:  1.70E+3nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232673(CHEMBL4061189)
Affinity DataKi:  3.69E+3nMAssay Description:Displacement of [3H]-5-CT from 5-HT7b receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232674(CHEMBL4068850)
Affinity DataKi:  4.29E+3nMAssay Description:Displacement of [3H]-Raclopride from D2L receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232667(CHEMBL4060194)
Affinity DataKi:  4.35E+3nMAssay Description:Displacement of [3H]-Raclopride from D2L receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232669(CHEMBL4079631)
Affinity DataKi:  5.16E+3nMAssay Description:Displacement of [3H]-Raclopride from D2L receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232666(CHEMBL4083059)
Affinity DataKi:  5.97E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232673(CHEMBL4061189)
Affinity DataKi:  6.70E+3nMAssay Description:Displacement of [3H]-Raclopride from D2L receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232671(CHEMBL4096141)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-Raclopride from D2L receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232671(CHEMBL4096141)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-5-CT from 5-HT7b receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232668(CHEMBL4103891)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232668(CHEMBL4103891)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-Raclopride from D2L receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232674(CHEMBL4068850)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-5-CT from 5-HT7b receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232674(CHEMBL4068850)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232670(CHEMBL4088416)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232671(CHEMBL4096141)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232672(CHEMBL4090862)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232668(CHEMBL4103891)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-5-CT from 5-HT7b receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232669(CHEMBL4079631)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-5-CT from 5-HT7b receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232667(CHEMBL4060194)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-5-CT from 5-HT7b receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232670(CHEMBL4088416)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-5-CT from 5-HT7b receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232672(CHEMBL4090862)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-5-CT from 5-HT7b receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232670(CHEMBL4088416)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-Raclopride from D2L receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232672(CHEMBL4090862)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-Raclopride from D2L receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232672(CHEMBL4090862)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232671(CHEMBL4096141)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232670(CHEMBL4088416)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232673(CHEMBL4061189)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232669(CHEMBL4079631)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50232667(CHEMBL4060194)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed