Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50001156
TargetProteasome subunit beta type-1(Human)
Hirosaki University

Curated by ChEMBL
LigandPNGBDBM50270495(CHEMBL4126890)
Affinity DataIC50: 1.73E+4nMAssay Description:Inhibition of human erythrocyte 20s proteasome caspase-like activity using Z-LLE-MCA as substrate pretreated for 10 mins followed by substrate additi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Hirosaki University

Curated by ChEMBL
LigandPNGBDBM50270495(CHEMBL4126890)
Affinity DataIC50: 1.85E+4nMAssay Description:Inhibition of human erythrocyte 20s proteasome chymotrypsin-like activity using Suc-LLVY-MCA as substrate pretreated for 10 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2020
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Hirosaki University

Curated by ChEMBL
LigandPNGBDBM50270495(CHEMBL4126890)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human erythrocyte 20s proteasome trypsin-like activity using Boc-LRR-MCA as substrate pretreated for 10 mins followed by substrate addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2020
Entry Details Article
PubMed