Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 50000033
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239459(CHEMBL4074929)
Affinity DataIC50: 30nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239465(CHEMBL4080525 | US11274074, Control [Ani9])
Affinity DataIC50: 77nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 20 mins followed by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239467(CHEMBL4086165)
Affinity DataIC50: 80nMAssay Description:Inhibition of TMEM16A (unknown origin) expressed in Xenopus laevis oocytes at -60 mV holding potential by voltage-clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239459(CHEMBL4074929)
Affinity DataIC50: 83nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239465(CHEMBL4080525 | US11274074, Control [Ani9])
Affinity DataIC50: 110nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239433(CHEMBL3134585)
Affinity DataIC50: 130nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239428(CHEMBL4104024)
Affinity DataIC50: 150nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239446(CHEMBL4069503)
Affinity DataIC50: 170nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239457(CHEMBL4071143)
Affinity DataIC50: 180nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239447(CHEMBL4090522)
Affinity DataIC50: 220nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239457(CHEMBL4071143)
Affinity DataIC50: 230nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239470(CHEMBL4095338)
Affinity DataIC50: 230nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239461(CHEMBL4074900)
Affinity DataIC50: 230nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239426(CHEMBL1444023)
Affinity DataIC50: 260nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239433(CHEMBL3134585)
Affinity DataIC50: 300nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239438(CHEMBL4099581)
Affinity DataIC50: 320nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239469(CHEMBL4091961)
Affinity DataIC50: 370nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239475(CHEMBL4082703)
Affinity DataIC50: 370nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239458(CHEMBL4095365)
Affinity DataIC50: 380nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239457(CHEMBL4071143)
Affinity DataIC50: 400nMAssay Description:Inhibition of human TMEM16B expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239459(CHEMBL4074929)
Affinity DataIC50: 400nMAssay Description:Inhibition of human TMEM16B expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239426(CHEMBL1444023)
Affinity DataIC50: 420nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239463(CHEMBL4087641)
Affinity DataIC50: 450nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239448(CHEMBL4080209)
Affinity DataIC50: 490nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239464(CHEMBL4085154)
Affinity DataIC50: 600nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239428(CHEMBL4104024)
Affinity DataIC50: 600nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239439(CHEMBL4083154)
Affinity DataIC50: 660nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239430(CHEMBL4096263)
Affinity DataIC50: 700nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239464(CHEMBL4085154)
Affinity DataIC50: 730nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239462(CHEMBL4066286)
Affinity DataIC50: 840nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239460(CHEMBL4103095)
Affinity DataIC50: 925nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239466(CHEMBL1299863)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239428(CHEMBL4104024)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human TMEM16B expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239436(CHEMBL4087045)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239478(CHEMBL4090401)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239472(CHEMBL4072679)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239456(CHEMBL4081693)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239437(CHEMBL4104905)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239443(CHEMBL4091843)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239450(CHEMBL4059811)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239464(CHEMBL4085154)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human TMEM16B expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-2(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239426(CHEMBL1444023)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human TMEM16B expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239476(CHEMBL4098234)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239467(CHEMBL4086165)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239431(CHEMBL4069000)
Affinity DataIC50: 1.88E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239432(CHEMBL4104747)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239455(CHEMBL4099708)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239435(CHEMBL4059668)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239474(CHEMBL4060277)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
TargetAnoctamin-1(Human)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239449(CHEMBL4088086)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2019
Entry Details Article
PubMed
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