Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50000542
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252992(CHEMBL4100496)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252998(CHEMBL4105008)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252992(CHEMBL4100496)
Affinity DataIC50: 0.190nMAssay Description:Inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252993(CHEMBL4073678)
Affinity DataIC50: 0.210nMAssay Description:Inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252997(CHEMBL4098116)
Affinity DataIC50: 0.280nMAssay Description:Inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252996(CHEMBL4097972)
Affinity DataIC50: 0.290nMAssay Description:Inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252994(CHEMBL4082551)
Affinity DataIC50: 0.290nMAssay Description:Inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252993(CHEMBL4073678)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252996(CHEMBL4097972)
Affinity DataIC50: 0.390nMAssay Description:Inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252995(CHEMBL4075535)
Affinity DataIC50: 0.410nMAssay Description:Inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50253005(CHEMBL4076887)
Affinity DataIC50: 0.450nMAssay Description:Inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50253004(CHEMBL4072122)
Affinity DataIC50: 0.470nMAssay Description:Inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252991(CHEMBL4064130)
Affinity DataIC50: 0.530nMAssay Description:Inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50253004(CHEMBL4072122)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252991(CHEMBL4064130)
Affinity DataIC50: 0.570nMAssay Description:Inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252998(CHEMBL4105008)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252995(CHEMBL4075535)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252992(CHEMBL4100496)
Affinity DataKi:  0.120nMAssay Description:Competitive inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252993(CHEMBL4073678)
Affinity DataKi:  0.120nMAssay Description:Non-competitive inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Linew...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252992(CHEMBL4100496)
Affinity DataKi:  0.270nMAssay Description:Competitive inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252996(CHEMBL4097972)
Affinity DataKi:  0.370nMAssay Description:Competitive inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252991(CHEMBL4064130)
Affinity DataKi:  0.610nMAssay Description:Competitive inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252994(CHEMBL4082551)
Affinity DataKi:  0.630nMAssay Description:Non-competitive inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Linew...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252998(CHEMBL4105008)
Affinity DataKi:  0.640nMAssay Description:Competitive inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252996(CHEMBL4097972)
Affinity DataKi:  0.660nMAssay Description:Competitive inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50253004(CHEMBL4072122)
Affinity DataKi:  0.660nMAssay Description:Competitive inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50253005(CHEMBL4076887)
Affinity DataKi:  0.690nMAssay Description:Competitive inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252991(CHEMBL4064130)
Affinity DataKi:  0.770nMAssay Description:Competitive inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252993(CHEMBL4073678)
Affinity DataKi:  0.880nMAssay Description:Competitive inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252997(CHEMBL4098116)
Affinity DataKi:  0.900nMAssay Description:Competitive inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50253004(CHEMBL4072122)
Affinity DataKi:  0.900nMAssay Description:Non-competitive inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Linew...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252998(CHEMBL4105008)
Affinity DataKi:  1.10nMAssay Description:Competitive inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252995(CHEMBL4075535)
Affinity DataKi:  5.10nMAssay Description:Competitive inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50252995(CHEMBL4075535)
Affinity DataKi:  6.20nMAssay Description:Competitive inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by Lineweave...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  8.90nMAssay Description:Inhibition of carbonic anhydrase-1 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 2(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  11nMAssay Description:Inhibition of carbonic anhydrase-2 in human erythrocyte membranes assessed as reduction in H+ release using CO2 as substrate by bromine thymol blue i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)