Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50000557
TargetHypoxia-inducible factor 1-alpha(Human)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50253289(CHEMBL4090212)
Affinity DataIC50: 600nMAssay Description:Inhibition of hypoxia-induced HIF1alpha (unknown origin) transcriptional activity expressed in human HCT116 cells by HRE luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50253288(CHEMBL4074474)
Affinity DataIC50: 870nMAssay Description:Inhibition of hypoxia-induced HIF1alpha (unknown origin) transcriptional activity expressed in human HCT116 cells by HRE luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50253276(CHEMBL4101212)
Affinity DataIC50: 940nMAssay Description:Inhibition of hypoxia-induced HIF1alpha (unknown origin) transcriptional activity expressed in human HCT116 cells by HRE luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50253294(CHEMBL4068303)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of hypoxia-induced HIF1alpha (unknown origin) transcriptional activity expressed in human HCT116 cells by HRE luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50253292(CHEMBL4098915)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of hypoxia-induced HIF1alpha (unknown origin) transcriptional activity expressed in human HCT116 cells by HRE luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50253291(CHEMBL4073157)
Affinity DataIC50: 4.52E+3nMAssay Description:Inhibition of hypoxia-induced HIF1alpha (unknown origin) transcriptional activity expressed in human HCT116 cells by HRE luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50253295(CHEMBL4080129)
Affinity DataIC50: 9.16E+3nMAssay Description:Inhibition of hypoxia-induced HIF1alpha (unknown origin) transcriptional activity expressed in human HCT116 cells by HRE luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50253290(CHEMBL4094550)
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibition of hypoxia-induced HIF1alpha (unknown origin) transcriptional activity expressed in human HCT116 cells by HRE luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2019
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50253293(CHEMBL4095572)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of hypoxia-induced HIF1alpha (unknown origin) transcriptional activity expressed in human HCT116 cells by HRE luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2019
Entry Details Article
PubMed