Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50001100
LigandPNGBDBM50243040(CHEMBL4065068)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to TACE catalytic domain (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed
LigandPNGBDBM50269406(CHEMBL4099646)
Affinity DataIC50: 61nMAssay Description:Inhibition of TACE in human whole blood assessed as inhibition of LPS-stimulated TNFalpha production pretreated for 1 hr followed by LPS stimulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed
LigandPNGBDBM50269407(CHEMBL4099281)
Affinity DataIC50: 92nMAssay Description:Inhibition of TACE in human whole blood assessed as inhibition of LPS-stimulated TNFalpha production pretreated for 1 hr followed by LPS stimulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed
LigandPNGBDBM50269399(CHEMBL4076728)
Affinity DataIC50: 104nMAssay Description:Inhibition of TACE in human whole blood assessed as inhibition of LPS-stimulated TNFalpha production pretreated for 1 hr followed by LPS stimulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed
LigandPNGBDBM50269400(CHEMBL4077272)
Affinity DataIC50: 141nMAssay Description:Inhibition of TACE in human whole blood assessed as inhibition of LPS-stimulated TNFalpha production pretreated for 1 hr followed by LPS stimulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed
LigandPNGBDBM50269408(CHEMBL4102424)
Affinity DataIC50: 156nMAssay Description:Inhibition of TACE in human whole blood assessed as inhibition of LPS-stimulated TNFalpha production pretreated for 1 hr followed by LPS stimulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed
LigandPNGBDBM50269404(CHEMBL4085841)
Affinity DataIC50: 176nMAssay Description:Inhibition of TACE in human whole blood assessed as inhibition of LPS-stimulated TNFalpha production pretreated for 1 hr followed by LPS stimulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed
LigandPNGBDBM50269401(CHEMBL4077298)
Affinity DataIC50: 178nMAssay Description:Inhibition of TACE in human whole blood assessed as inhibition of LPS-stimulated TNFalpha production pretreated for 1 hr followed by LPS stimulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed
LigandPNGBDBM50269397(CHEMBL4074184)
Affinity DataIC50: 281nMAssay Description:Inhibition of TACE in human whole blood assessed as inhibition of LPS-stimulated TNFalpha production pretreated for 1 hr followed by LPS stimulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed
LigandPNGBDBM50269402(CHEMBL4098911)
Affinity DataIC50: 282nMAssay Description:Inhibition of TACE in human whole blood assessed as inhibition of LPS-stimulated TNFalpha production pretreated for 1 hr followed by LPS stimulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed
LigandPNGBDBM50243040(CHEMBL4065068)
Affinity DataIC50: 287nMAssay Description:Inhibition of TACE in human whole blood assessed as inhibition of LPS-stimulated TNFalpha production pretreated for 1 hr followed by LPS stimulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed
LigandPNGBDBM50269403(CHEMBL4080126)
Affinity DataIC50: 339nMAssay Description:Inhibition of TACE in human whole blood assessed as inhibition of LPS-stimulated TNFalpha production pretreated for 1 hr followed by LPS stimulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed
LigandPNGBDBM50269405(CHEMBL4068636)
Affinity DataIC50: 560nMAssay Description:Inhibition of TACE in human whole blood assessed as inhibition of LPS-stimulated TNFalpha production pretreated for 1 hr followed by LPS stimulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed
LigandPNGBDBM50269398(CHEMBL4089626)
Affinity DataIC50: 7.15E+3nMAssay Description:Inhibition of TACE in human whole blood assessed as inhibition of LPS-stimulated TNFalpha production pretreated for 1 hr followed by LPS stimulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2020
Entry Details Article
PubMed