Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50002293
TargetGlutamate receptor 2(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50456718(CHEMBL4208162)
Affinity DataKi:  1.71E+3nMAssay Description:Displacement of [3H]AMPA from rat GluA2(R) receptor flip isoform expressed in sf9 insect cell membranes by TopCount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamate receptor 2(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50456718(CHEMBL4208162)
Affinity DataKi:  1.74E+3nMAssay Description:Displacement of [3H]AMPA from rat GluA2(Q) receptor flop isoform by TopCount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamate receptor 3(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50456718(CHEMBL4208162)
Affinity DataKi:  7.01E+3nMAssay Description:Displacement of [3H]AMPA from rat GluA3 receptor flip isoform expressed in sf9 insect cell membranes by TopCount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamate receptor 2(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50456716(CHEMBL4207628)
Affinity DataKi:  1.84E+4nMAssay Description:Displacement of [3H]AMPA from rat GluA2(R) receptor flip isoform expressed in sf9 insect cell membranes by TopCount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamate receptor 2(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50456717(CHEMBL4212533)
Affinity DataKi:  2.07E+4nMAssay Description:Displacement of [3H]AMPA from rat GluA2(R) receptor flip isoform expressed in sf9 insect cell membranes by TopCount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamate receptor 2(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50456719(CHEMBL4216018)
Affinity DataKi:  2.19E+4nMAssay Description:Displacement of [3H]AMPA from rat GluA2(R) receptor flip isoform expressed in sf9 insect cell membranes by TopCount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamate receptor 2(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50456720(CHEMBL4211059)
Affinity DataKi:  4.08E+4nMAssay Description:Displacement of [3H]AMPA from rat GluA2(R) receptor flip isoform expressed in sf9 insect cell membranes by TopCount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamate receptor 3(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50456716(CHEMBL4207628)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AMPA from rat GluA3 receptor flip isoform expressed in sf9 insect cell membranes by TopCount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamate receptor 3(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50456719(CHEMBL4216018)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AMPA from rat GluA3 receptor flip isoform expressed in sf9 insect cell membranes by TopCount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamate receptor 3(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50456717(CHEMBL4212533)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AMPA from rat GluA3 receptor flip isoform expressed in sf9 insect cell membranes by TopCount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamate receptor 2(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50456721(CHEMBL4215471)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AMPA from rat GluA2(R) receptor flip isoform expressed in sf9 insect cell membranes by TopCount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamate receptor 3(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50456720(CHEMBL4211059)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AMPA from rat GluA3 receptor flip isoform expressed in sf9 insect cell membranes by TopCount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutamate receptor 3(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50456721(CHEMBL4215471)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AMPA from rat GluA3 receptor flip isoform expressed in sf9 insect cell membranes by TopCount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed