Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50000785
TargetDiacylglycerol O-acyltransferase 1(Human)
Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50260380(CHEMBL4092694)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of recombinant full length human DGAT1 expressed in Sf9 insect cells using 1,2-didecanoyl-sn-glycerol as substrate after 60 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50260377(CHEMBL4096065)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of recombinant full length human DGAT1 expressed in Sf9 insect cells using 1,2-didecanoyl-sn-glycerol as substrate after 60 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM20716((1R,2R)-2-[(4-{4-[(phenylcarbamoyl)amino]phenyl}ph...)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of recombinant full length human DGAT1 expressed in Sf9 insect cells using 1,2-didecanoyl-sn-glycerol as substrate after 60 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50260376(CHEMBL4095138)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of recombinant full length human DGAT1 expressed in Sf9 insect cells using 1,2-didecanoyl-sn-glycerol as substrate after 60 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50260382(CHEMBL4068759)
Affinity DataIC50: 8.80nMAssay Description:Inhibition of recombinant full length human DGAT1 expressed in Sf9 insect cells using 1,2-didecanoyl-sn-glycerol as substrate after 60 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50260374(CHEMBL4066063)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant full length human DGAT1 expressed in Sf9 insect cells using 1,2-didecanoyl-sn-glycerol as substrate after 60 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50260381(CHEMBL4074675)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant full length human DGAT1 expressed in Sf9 insect cells using 1,2-didecanoyl-sn-glycerol as substrate after 60 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50260379(CHEMBL4099177)
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant full length human DGAT1 expressed in Sf9 insect cells using 1,2-didecanoyl-sn-glycerol as substrate after 60 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50260373(CHEMBL4065011)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant full length human DGAT1 expressed in Sf9 insect cells using 1,2-didecanoyl-sn-glycerol as substrate after 60 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50260375(CHEMBL4087443)
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant full length human DGAT1 expressed in Sf9 insect cells using 1,2-didecanoyl-sn-glycerol as substrate after 60 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50260378(CHEMBL4075629)
Affinity DataIC50: 38nMAssay Description:Inhibition of recombinant full length human DGAT1 expressed in Sf9 insect cells using 1,2-didecanoyl-sn-glycerol as substrate after 60 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50260371(CHEMBL4084613)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant full length human DGAT1 expressed in Sf9 insect cells using 1,2-didecanoyl-sn-glycerol as substrate after 60 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Xinxiang Medical University

Curated by ChEMBL
LigandPNGBDBM50260372(CHEMBL4102892)
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant full length human DGAT1 expressed in Sf9 insect cells using 1,2-didecanoyl-sn-glycerol as substrate after 60 mins in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/13/2020
Entry Details Article
PubMed