Compile Data Set for Download or QSAR
Report error Found 309 Enz. Inhib. hit(s) with all data for entry = 50002294
Target5-hydroxytryptamine receptor 5A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456745(CHEMBL4207302)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT5A receptor expressed in Flp-In CHO cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456743(CHEMBL4217810)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT5A receptor expressed in Flp-In CHO cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456743(CHEMBL4217810)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-GR65630 from human 5-HT3 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456743(CHEMBL4217810)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]5-CT from human 5-HT1D receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456743(CHEMBL4217810)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A (unknown origin) receptor after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456726(CHEMBL4218231)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A (unknown origin) receptor after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456745(CHEMBL4207302)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]5-CT from human 5-HT1B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456726(CHEMBL4218231)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT7A receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456743(CHEMBL4217810)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]5-CT from human 5-HT1B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456726(CHEMBL4218231)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456743(CHEMBL4217810)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1E(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456743(CHEMBL4217810)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]5-HT from human 5-HT1E receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456745(CHEMBL4207302)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A (unknown origin) receptor after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456726(CHEMBL4218231)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-GR65630 from human 5-HT3 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456743(CHEMBL4217810)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-Mesulergine from human 5-HT2C receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456745(CHEMBL4207302)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]5-CT from human 5-HT1D receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456726(CHEMBL4218231)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]5-CT from human 5-HT1D receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456743(CHEMBL4217810)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT7A receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456726(CHEMBL4218231)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]5-CT from human 5-HT1B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 5A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456726(CHEMBL4218231)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT5A receptor expressed in Flp-In CHO cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1E(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456726(CHEMBL4218231)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]5-HT from human 5-HT1E receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456745(CHEMBL4207302)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1E(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456745(CHEMBL4207302)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]5-HT from human 5-HT1E receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456745(CHEMBL4207302)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT7A receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456745(CHEMBL4207302)
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-GR65630 from human 5-HT3 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456728(CHEMBL4212246)
Affinity DataEC50:  29nMAssay Description:Partial agonist activity at 5-HT1B receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456734(CHEMBL4212435)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]-LSD from human 5-HT2B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456741(CHEMBL4204036)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]-GR65630 from human 5-HT3 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456740(CHEMBL4205064)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]-LSD from human 5-HT2B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456727(CHEMBL4209942)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]-LSD from human 5-HT2B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456745(CHEMBL4207302)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-LSD from human 5-HT2B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456734(CHEMBL4212435)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]-Mesulergine from human 5-HT2C receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456735(CHEMBL4204576)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-GR65630 from human 5-HT3 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456732(CHEMBL4207355)
Affinity DataEC50:  180nMAssay Description:Partial agonist activity at 5-HT1B receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456734(CHEMBL4212435)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]-GR65630 from human 5-HT3 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456742(CHEMBL4208914)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A (unknown origin) receptor after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456739(CHEMBL4208376)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A (unknown origin) receptor after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456737(CHEMBL4216860)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A (unknown origin) receptor after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456735(CHEMBL4204576)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]-LSD from human 5-HT2B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456743(CHEMBL4217810)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]-LSD from human 5-HT2B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50335603(Pulicatin A | CHEMBL1651095)
Affinity DataKi:  510nMAssay Description:Displacement of [3H]-LSD from human 5-HT2B receptor expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456724(CHEMBL4207529)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]5-CT from human 5-HT1D receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456726(CHEMBL4218231)
Affinity DataKi:  620nMAssay Description:Displacement of [3H]-LSD from human 5-HT2B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456741(CHEMBL4204036)
Affinity DataKi:  690nMAssay Description:Displacement of [3H]-LSD from human 5-HT2B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456741(CHEMBL4204036)
Affinity DataKi:  750nMAssay Description:Displacement of [3H]-Mesulergine from human 5-HT2C receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456727(CHEMBL4209942)
Affinity DataKi:  770nMAssay Description:Displacement of [3H]-Mesulergine from human 5-HT2C receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456735(CHEMBL4204576)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]5-CT from human 5-HT1D receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456734(CHEMBL4212435)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456736(CHEMBL4210787)
Affinity DataKi:  810nMAssay Description:Displacement of [3H]-LSD from human 5-HT2B receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of The Philippines

Curated by ChEMBL
LigandPNGBDBM50456737(CHEMBL4216860)
Affinity DataKi:  820nMAssay Description:Displacement of [3H]-Mesulergine from human 5-HT2C receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
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