Report error Found 309 Enz. Inhib. hit(s) with all data for entry = 50002294
Affinity DataEC50: 180nMAssay Description:Partial agonist activity at 5-HT1B receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataEC50: 29nMAssay Description:Partial agonist activity at 5-HT1B receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Antagonist activity at 5-HT1B receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Antagonist activity at 5-HT1B receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+3nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:Antagonist activity at 5-HT2C receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT1A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT1A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT7A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT7A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT4 receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT1D receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT1D receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT2C receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT2C receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT1A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT1A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT1A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT1A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT1A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT4 receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT7A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT1D receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT1A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at 5-HT1A receptor (unknown origin) by Tango assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Antagonist activity at 5-HT2A receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) by calcium release assayMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A (unknown origin) receptor after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT5A receptor expressed in Flp-In CHO cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT7A receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT5A receptor expressed in Flp-In CHO cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-LSD from human 5-HT5A receptor expressed in Flp-In CHO cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-GR65630 from human 5-HT3 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-GR65630 from human 5-HT3 receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]-Mesulergine from human 5-HT2C receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A (unknown origin) receptor after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]5-HT from human 5-HT1E receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]5-HT from human 5-HT1E receptor expressed in HEK cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]5-CT from human 5-HT1D receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H]5-CT from human 5-HT1D receptor expressed in HEKT cells after 90 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair












