Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50000117
TargetGlucagon-like peptide 1 receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50121394(CHEMBL3616711)
Affinity DataEC50:  0.0230nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2019
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50152769(GLP-1(7-36)-NH2 | NH2-HAEGTFTSDVSSYLEGQAAKEFIAWLVK...)
Affinity DataEC50:  0.0440nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2019
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240819(CHEMBL4084119)
Affinity DataEC50:  0.0670nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2019
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240820(CHEMBL4073765)
Affinity DataEC50:  0.0680nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2019
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240823(CHEMBL4083273)
Affinity DataEC50:  0.118nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2019
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240824(CHEMBL4062410)
Affinity DataEC50:  0.148nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2019
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240821(CHEMBL4100575)
Affinity DataEC50:  0.221nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2019
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240825(CHEMBL4103967)
Affinity DataEC50:  0.522nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2019
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240822(CHEMBL4079706)
Affinity DataEC50:  0.547nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2019
Entry Details Article
PubMed
TargetAlbumin(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataKd:  700nMAssay Description:Binding affinity to human serum albuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAlbumin(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240510(CHEMBL898 | DIFLUNISAL)
Affinity DataKd:  3.00E+3nMAssay Description:Binding affinity to human serum albuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2019
Entry Details Article
PubMed