Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50001131
TargetAdenosine receptor A1(Bovine)
North-West University

Curated by ChEMBL
LigandPNGBDBM50120761(Cyclopentanecarboxylic acid (7-methyl-2-phenyl-imi...)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]CHA from A1 receptor in bovine cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
North-West University

Curated by ChEMBL
LigandPNGBDBM50120765(1-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CHA from A1 receptor in bovine cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
North-West University

Curated by ChEMBL
LigandPNGBDBM50120764(Cyclopentanecarboxylic acid (2,7-diphenyl-imidazo[...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]CHA from A1 receptor in bovine cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
North-West University

Curated by ChEMBL
LigandPNGBDBM50120760(Cyclohexanecarboxylic acid (7-methyl-2-phenyl-imid...)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]CHA from A1 receptor in bovine cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
North-West University

Curated by ChEMBL
LigandPNGBDBM50120754(Cyclohexylmethyl-(7-methyl-2-phenyl-imidazo[1,2-a]...)
Affinity DataKi:  231nMAssay Description:Displacement of [3H]CHA from A1 receptor in bovine cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
North-West University

Curated by ChEMBL
LigandPNGBDBM50120757(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-4-y...)
Affinity DataKi:  332nMAssay Description:Displacement of [3H]CHA from A1 receptor in bovine cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
North-West University

Curated by ChEMBL
LigandPNGBDBM50120753(N-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi:  855nMAssay Description:Displacement of [3H]CHA from A1 receptor in bovine cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269832(CHEMBL4065991)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membrane assessed as effect on GTP shift in presence of 100 uM GTPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269832(CHEMBL4065991)
Affinity DataKi:  2.06E+3nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269831(CHEMBL1807296)
Affinity DataKi:  3.90E+3nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269833(CHEMBL1807329)
Affinity DataKi:  5.53E+3nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269839(CHEMBL1807282)
Affinity DataKi:  7.61E+3nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269832(CHEMBL4065991)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269828(CHEMBL1807327)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269833(CHEMBL1807329)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269834(CHEMBL1807290)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269835(CHEMBL1303604)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50444540(CHEMBL1594316)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269836(CHEMBL1621581)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269836(CHEMBL1621581)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269837(CHEMBL377488)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269829(CHEMBL1807324)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269830(CHEMBL1807298)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269828(CHEMBL1807327)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269837(CHEMBL377488)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269831(CHEMBL1807296)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269838(CHEMBL1807293)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269839(CHEMBL1807282)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269840(CHEMBL4084890)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269841(CHEMBL1720835)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269829(CHEMBL1807324)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269834(CHEMBL1807290)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269838(CHEMBL1807293)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269830(CHEMBL1807298)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-NECA from A2A receptor in rat striatal membrane in presence of A1 receptor agonist N6-cyclopentyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269840(CHEMBL4084890)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269835(CHEMBL1303604)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50444540(CHEMBL1594316)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
North-West University

Curated by ChEMBL
LigandPNGBDBM50269841(CHEMBL1720835)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-DPCPX from A1 receptor in rat whole brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMed