Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50000120
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(6-(3-iodobenzylamino)-2-chloro-9H-pu...)
Affinity DataKi:  0.00483nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214981((2R,3R,4S)-2-(2-chloro-6-(3-chlorobenzylamino)-9H-...)
Affinity DataKi:  0.0102nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataKi:  0.0480nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50085048((S)-2-(2-benzoylphenylamino)-3-(4-(2-(methyl(pyrid...)
Affinity DataKi:  0.0497nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARgamma LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50099491(cid_3392731 | CHEMBL21241 | 2-(4-{2-[3-Cyclohexyl-...)
Affinity DataKi:  0.0541nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARalpha LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50180197((2S,3S,4R,5R)-5-(2-chloro-6-(3-iodobenzylamino)-9H...)
Affinity DataKi:  0.160nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304633(9-(5'-Cyclobutylaminocarbonyl-4'-thio-beta-D-ribof...)
Affinity DataKi:  0.170nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARgamma LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50252829((2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-9H-purin-9-...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50180197((2S,3S,4R,5R)-5-(2-chloro-6-(3-iodobenzylamino)-9H...)
Affinity DataKi:  0.380nMAssay Description:Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304635(9-(5'-Ethylaminocarbonyl-4-thio-beta-D-ribofuranos...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM21221(2-Cl-IB-MECA | CHEMBL431733 | C-IBzA-MU | 2-chloro...)
Affinity DataKi:  0.430nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214980((2R,3R,4S)-2-(2-chloro-6-(2-chlorobenzylamino)-9H-...)
Affinity DataKi:  0.620nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304633(9-(5'-Cyclobutylaminocarbonyl-4'-thio-beta-D-ribof...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM21221(2-Cl-IB-MECA | CHEMBL431733 | C-IBzA-MU | 2-chloro...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A3(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50252757((2R,3R,4S)-2-(6-(3-Iodobenzylamino)-9H-purin-9-yl)...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214981((2R,3R,4S)-2-(2-chloro-6-(3-chlorobenzylamino)-9H-...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304639(9-(5'-Cyclopropylmethylaminocarbonyl-4'-thio-beta-...)
Affinity DataKi:  1.80nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARgamma LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50118812(CHEMBL119709 | (3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-io...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A3(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304639(9-(5'-Cyclopropylmethylaminocarbonyl-4'-thio-beta-...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM21221(2-Cl-IB-MECA | CHEMBL431733 | C-IBzA-MU | 2-chloro...)
Affinity DataKi:  2.20nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARgamma LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304639(9-(5'-Cyclopropylmethylaminocarbonyl-4'-thio-beta-...)
Affinity DataKi:  2.40nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50252829((2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-9H-purin-9-...)
Affinity DataKi:  2.5nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304633(9-(5'-Cyclobutylaminocarbonyl-4'-thio-beta-D-ribof...)
Affinity DataKi:  2.60nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304637(9-(5'-Cyclopropylaminocarbonyl-4'-thio-beta-D-ribo...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304637(9-(5'-Cyclopropylaminocarbonyl-4'-thio-beta-D-ribo...)
Affinity DataKi:  3nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304635(9-(5'-Ethylaminocarbonyl-4-thio-beta-D-ribofuranos...)
Affinity DataKi:  3.20nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARdelta LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(6-(3-iodobenzylamino)-2-chloro-9H-pu...)
Affinity DataKi:  3.40nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARgamma LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(6-(3-iodobenzylamino)-2-chloro-9H-pu...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50180197((2S,3S,4R,5R)-5-(2-chloro-6-(3-iodobenzylamino)-9H...)
Affinity DataKi:  4.60nMAssay Description:Displacement of Fluormone-Pan-PPAR Green from human GST-tagged PPARgamma LBD by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304635(9-(5'-Ethylaminocarbonyl-4-thio-beta-D-ribofuranos...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]CCPA from human A1 receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304637(9-(5'-Cyclopropylaminocarbonyl-4'-thio-beta-D-ribo...)
Affinity DataKi:  9.30nMAssay Description:Displacement of [3H]CCPA from human A1 receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304637(9-(5'-Cyclopropylaminocarbonyl-4'-thio-beta-D-ribo...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50252829((2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-9H-purin-9-...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CCPA from human A1 receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304633(9-(5'-Cyclobutylaminocarbonyl-4'-thio-beta-D-ribof...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]CCPA from human A1 receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214980((2R,3R,4S)-2-(2-chloro-6-(2-chlorobenzylamino)-9H-...)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50118812(CHEMBL119709 | (3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-io...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]CCPA from human A1 receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304635(9-(5'-Ethylaminocarbonyl-4-thio-beta-D-ribofuranos...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304633(9-(5'-Cyclobutylaminocarbonyl-4'-thio-beta-D-ribof...)
Affinity DataKi:  122nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304639(9-(5'-Cyclopropylmethylaminocarbonyl-4'-thio-beta-...)
Affinity DataKi:  159nMAssay Description:Displacement of [3H]CCPA from human A1 receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50180197((2S,3S,4R,5R)-5-(2-chloro-6-(3-iodobenzylamino)-9H...)
Affinity DataKi:  193nMAssay Description:Displacement of [3H]CCPA from human A1 receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM21221(2-Cl-IB-MECA | CHEMBL431733 | C-IBzA-MU | 2-chloro...)
Affinity DataKi:  222nMAssay Description:Displacement of [3H]CCPA from human A1 receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50180197((2S,3S,4R,5R)-5-(2-chloro-6-(3-iodobenzylamino)-9H...)
Affinity DataKi:  223nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(6-(3-iodobenzylamino)-2-chloro-9H-pu...)
Affinity DataKi:  341nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50252757((2R,3R,4S)-2-(6-(3-Iodobenzylamino)-9H-purin-9-yl)...)
Affinity DataKi:  440nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50252829((2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-9H-purin-9-...)
Affinity DataKi:  475nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50252757((2R,3R,4S)-2-(6-(3-Iodobenzylamino)-9H-purin-9-yl)...)
Affinity DataKi:  860nMAssay Description:Displacement of [3H]CCPA from human A1 receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214980((2R,3R,4S)-2-(2-chloro-6-(2-chlorobenzylamino)-9H-...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50304639(9-(5'-Cyclopropylmethylaminocarbonyl-4'-thio-beta-...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(6-(3-iodobenzylamino)-2-chloro-9H-pu...)
Affinity DataKi:  2.49E+3nMAssay Description:Displacement of [3H]CCPA from human A1 receptor expressed in CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Sahmyook University

Curated by ChEMBL
LigandPNGBDBM50118812(CHEMBL119709 | (3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-io...)
Affinity DataKi:  2.91E+3nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
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