Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50001956
TargetHeparanase(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50450965(CHEMBL4204865)
Affinity DataIC50: 660nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHeparanase(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50450963(CHEMBL4218441)
Affinity DataIC50: 860nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHeparanase(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50450967(CHEMBL4215493)
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHeparanase(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50450964(CHEMBL4211674)
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHeparanase(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50450962(CHEMBL4203220)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHeparanase(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50450960(CHEMBL4206187)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHeparanase(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50450961(CHEMBL4213074)
Affinity DataIC50: 5.64E+3nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHeparanase(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50450966(CHEMBL4210546)
Affinity DataIC50: 8.53E+3nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHeparanase(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179360(CHEMBL3040216)
Affinity DataIC50: 2.66E+4nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHeparanase(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50179360(CHEMBL3040216)
Affinity DataKi:  4.80E+4nMAssay Description:Inhibition of mouse B16-BL6 cells derived heparanase using [3H]HS as substrate after 6 hrs by size exclusion chromatography based liquid scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed