Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50048752
LigandPNGBDBM50226801(CHEMBL7707)
Affinity DataKi:  0.550nMAssay Description:Binding affinity for alpha-2 adrenergic receptor in rat cortex using [3H]rauwolscine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226802(CHEMBL7186)
Affinity DataKi:  6.5nMAssay Description:Binding affinity for alpha-2 adrenergic receptor in rat cortex using [3H]rauwolscine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50019729(A-54741 | CHEMBL7169 | (S)-5-(4,5-Dihydro-1H-imida...)
Affinity DataKi:  28nMAssay Description:Binding affinity for alpha-2 adrenergic receptor in rat cortex using [3H]rauwolscine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50225285(CHEBI:3757 | Catapres | Catapres-Tts-1 | Catapres-...)
Affinity DataKi:  30nMAssay Description:Binding affinity for alpha-2 adrenergic receptor in rat cortex using [3H]rauwolscine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50029051(4-[(1R)-2-amino-1-hydroxyethyl]benzene-1,2-diol | ...)
Affinity DataKi:  37nMAssay Description:Binding affinity for alpha-2 adrenergic receptor in rat cortex using [3H]rauwolscine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50029051(4-[(1R)-2-amino-1-hydroxyethyl]benzene-1,2-diol | ...)
Affinity DataKi:  390nMAssay Description:Binding affinity for alpha-1 adrenergic receptor in rat liver using [3H]prazosin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226802(CHEMBL7186)
Affinity DataKi:  400nMAssay Description:Binding affinity for alpha-1 adrenergic receptor in rat liver using [3H]prazosin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50225285(CHEBI:3757 | Catapres | Catapres-Tts-1 | Catapres-...)
Affinity DataKi:  520nMAssay Description:Binding affinity for alpha-1 adrenergic receptor in rat liver using [3H]prazosin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226801(CHEMBL7707)
Affinity DataKi:  523nMAssay Description:Binding affinity for alpha-1 adrenergic receptor in rat liver using [3H]prazosin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50019729(A-54741 | CHEMBL7169 | (S)-5-(4,5-Dihydro-1H-imida...)
Affinity DataKi:  817nMAssay Description:Binding affinity for alpha-1 adrenergic receptor in rat liver using [3H]prazosin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed