Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50018902
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613723(CHEMBL5268330)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613719(CHEMBL5281165)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613721(CHEMBL5275547)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCytochrome P450 1A2(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCytochrome P450 2C19(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCytochrome P450 2C9(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCytochrome P450 2D6(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCytochrome P450 3A4(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613720(CHEMBL5283073)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613716(CHEMBL5283476)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613718(CHEMBL5286709)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613726(CHEMBL5272922)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613724(CHEMBL5268485)
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613722(CHEMBL5289708)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50613717(CHEMBL5276028)
Affinity DataIC50: 1.13E+5nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed