Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50000140
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50241432(CHEMBL4061049)
Affinity DataEC50:  4.00E+4nMAssay Description:Partial agonist activity at human alpha7 nAChR expressed in Xenopus laevis oocytes assessed as induction of maximum current response administered for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50241434(CHEMBL3747954)
Affinity DataEC50:  2.21E+5nMAssay Description:Partial agonist activity at human alpha7 nAChR expressed in Xenopus laevis oocytes assessed as induction of maximum current response administered for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50241437(CHEMBL4082927)
Affinity DataIC50: 1.15E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response admini...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50241432(CHEMBL4061049)
Affinity DataIC50: 5.10E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50241434(CHEMBL3747954)
Affinity DataIC50: 5.50E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response admini...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50241432(CHEMBL4061049)
Affinity DataIC50: 7.30E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response admini...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2019
Entry Details Article
PubMed